SCHEMBL29329368

SCHEMBL29329368

N#Cc1cc(OCCc2cccc(C(F)(F)F)c2)cc(Nc2ccc3cc[nH]c3c2)n1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
PRKCQ Q04759 3/20 0.37
IDH1 O75874 1/20 0.37
KIF11 P52732 1/20 0.36
MET P08581 1/20 0.36
GALR2 O43603 1/20 0.35
TTBK1 Q5TCY1 2/20 0.35
AURKA O14965 1/20 0.35
CDK8 P49336 1/20 0.35
GPR52 Q9Y2T5 1/20 0.35
SLC2A1 P11166 1/20 0.35
CTSS P25774 1/20 0.34
NR3C2 P08235 1/20 0.34
TTBK2 Q6IQ55 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29329869 0.92 ESR1 (0.42) ESR1SIRT2IDH1KIF11
SCHEMBL29330563 0.88 PRKCQ (0.39) ESR1SIRT2PRKCQMETSLC2A1
SCHEMBL29329290 0.87 PRKCQ (0.42) ESR1PRKCQMET
SCHEMBL29328815 0.87 MAOB (0.40) SIRT2PRKCQMET
SCHEMBL29329720 0.85 TTBK1 (0.46) ESR1PRKCQIDH1KIF11TTBK1
SCHEMBL29329365 0.85 MET (0.40) ESR1PRKCQMET
SCHEMBL29330428 0.84 ESR1 (0.42) ESR1PRKCQGALR2
SCHEMBL29329726 0.84 SYK (0.39) ESR1PRKCQMET
SCHEMBL29330026 0.83 SIRT2 (0.40) ESR1SIRT2PRKCQ
SCHEMBL29329867 0.82 PRKCQ (0.40) ESR1SIRT2PRKCQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024151919-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY IFM DUE, INC. (US) 2024-07-18 WO disclosed