Venglustat

Venglustat

SCHEMBL29358474

CC(C)(NC(=O)O[C@H]1CN2CCC1CC2)c1csc(-c2ccc(F)cc2)n1.O=C(O)CC(O)C(=O)O

nearest known ligand 0.83

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

UGCG

The experimentally established mechanism targets of Venglustat. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
UGCG known ✓ Q16739 1/20 0.83
NTMT1 Q9BV86 20/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Venglustat SCHEMBL31522597 1.00 NTMT1 (0.83) NTMT1UGCG
Venglustat SCHEMBL12615333 0.91 NTMT1 (1.00) NTMT1UGCG
Venglustat SCHEMBL29359568 0.91 NTMT1 (1.00) NTMT1UGCG
Venglustat SCHEMBL12615329 0.91 NTMT1 (1.00) NTMT1UGCG
Venglustat SCHEMBL19844439 0.91 NTMT1 (1.00) NTMT1UGCG
SCHEMBL19407265 0.84 NTMT1 (1.00) NTMT1UGCG
SCHEMBL18309554 0.83 NTMT1 (1.00) NTMT1UGCG
Malic Acid SCHEMBL23234120 0.81 NTMT1 (0.50) NTMT1UGCG
Malic Acid SCHEMBL17504472 0.80 NTMT1 (0.52) NTMT1UGCG
Malic Acid SCHEMBL17504470 0.80 NTMT1 (0.52) NTMT1UGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4626424-A1 VENGLUSTAT IN COMBINATION WITH A STRONG OR MODERATE INHIBITOR OF CYP3A4 GENZYME CORPORATION (US) 2025-10-08 EP claimed
WO-2024116127-A1 VENGLUSTAT IN COMBINATION WITH A STRONG OR MODERATE INHIBITOR OF CYP3A4 GENZYME CORPORATION (US) 2024-06-06 WO claimed
EP-4349408-A2 METHODS FOR TREATING PROTEINOPATHIES Genzyme Corporation (US) 2024-04-10 EP claimed
US-20240091208-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT GENZYME CORPORATION 2024-03-21 US claimed
US-11857512-B2 Pharmaceutical compositions comprising venglustat GENZYME CORPORATION (US) 2024-01-02 US claimed
EP-4185267-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT Genzyme Corporation (US) 2023-05-31 EP claimed
US-20220023272-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT GENZYME CORPORATION 2022-01-27 US claimed
WO-2022018695-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT GENZYME CORPORATION (US) 2022-01-27 WO claimed
WO-2025262570-A1 VENGLUSTAT AS AN INHIBITOR OF GLUCOSYLCERAMIDE SYNTHASE IN SUBJECTS HAVING HEPATIC IMPAIRMENT GENZYME CORPORATION (US) 2025-12-26 WO disclosed
US-20250354999-A1 BIOMARKERS OF LYSOSOMAL STORAGE DISEASE GENZYME CORP (US) 2025-11-20 US disclosed
EP-4626424-A1 VENGLUSTAT IN COMBINATION WITH A STRONG OR MODERATE INHIBITOR OF CYP3A4 GENZYME CORPORATION (US) 2025-10-08 EP disclosed
EP-4558828-A1 BIOMARKERS OF LYSOSOMAL STORAGE DISEASE GENZYME CORPORATION (US) 2025-05-28 EP disclosed
CN-119630967-A Biomarkers for lysosomal storage diseases 建新公司 2025-03-14 CN disclosed
WO-2024116127-A1 VENGLUSTAT IN COMBINATION WITH A STRONG OR MODERATE INHIBITOR OF CYP3A4 GENZYME CORPORATION (US) 2024-06-06 WO disclosed
EP-4185267-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT Genzyme Corporation (US) 2023-05-31 EP disclosed
US-20230067811-A1 MODULATING LYMPHATIC VESSELS IN NEUROLOGICAL DISEASE UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2023-03-02 US disclosed
EP-4093426-A1 MODULATING LYMPHATIC VESSELS IN NEUROLOGICAL DISEASE University of Virginia Patent Foundation (US) 2022-11-30 EP disclosed
US-20220152031-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GOLDFINCH BIO, INC. 2022-05-19 US disclosed
US-20220023272-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT GENZYME CORPORATION 2022-01-27 US disclosed
WO-2022018695-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT GENZYME CORPORATION (US) 2022-01-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220023272-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT SOST, SLC5A1, SLC10A6 UGCG 60/4885NTMT1 649/4885
US-20240091208-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING VENGLUSTAT SOST, SLC5A1, SLC10A6 UGCG 60/4885NTMT1 649/4885
US-20220152031-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GLS, ATP6V1B1, PDXK UGCG 1842/4885NTMT1 3179/4885
US-11857512-B2 Pharmaceutical compositions comprising venglustat SOST, SLC5A1, SLC10A6 UGCG 60/4885NTMT1 649/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.