Ifidancitinib

Ifidancitinib

SCHEMBL29360646

COc1cc(Nc2ncc(C)c(Nc3ccc4oc(=O)[nH]c4c3)n2)cc(C)c1F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 20/20 1.00
JAK3 P52333 20/20 1.00
JAK2 O60674 12/20 1.00
CYP1A2 P05177 2/20 1.00
TYK2 P29597 1/20 1.00
CYP3A4 P08684 9/20 0.83
SYK P43405 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ifidancitinib SCHEMBL342002 1.00 JAK1 (1.00) JAK1JAK3JAK2CYP1A2TYK2
Ifidancitinib SCHEMBL29609558 1.00 JAK1 (1.00) JAK1JAK3JAK2CYP1A2TYK2
Ifidancitinib SCHEMBL20767498 0.99 JAK1 (0.98) JAK1JAK3JAK2CYP1A2TYK2
Ifidancitinib SCHEMBL29358204 0.96 JAK1 (0.92) JAK1JAK3JAK2CYP1A2TYK2
Ifidancitinib SCHEMBL29358557 0.96 JAK1 (0.92) JAK1JAK3JAK2CYP1A2TYK2
Ifidancitinib SCHEMBL525194 0.96 JAK1 (0.92) JAK1JAK3JAK2CYP1A2TYK2
Ifidancitinib SCHEMBL525310 0.96 JAK1 (0.92) JAK1JAK3JAK2CYP1A2TYK2
Ifidancitinib SCHEMBL23356291 0.95 JAK1 (0.90) JAK1JAK3JAK2CYP1A2TYK2
SCHEMBL23356183 0.94 JAK1 (0.88) JAK1JAK3JAK2CYP1A2TYK2
SCHEMBL339570 0.94 JAK1 (0.88) JAK1JAK3JAK2CYP1A2TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12617805-B2 Codrug that disintegrates in intestine, preparation therefor, and use thereof ENNOVABIO (ZHEJIANG) PHARMACEUTICALS CO., LTD. (CN) 2026-05-05 US claimed
US-20250367113-A1 DRUG DELIVERY SYSTEM COMPRISING AN ANTI-INFLAMMATORY AGENT OR A SALT THEREOF FOR THE APPLICATION TO ESOPHAGEAL MUCOUS MEMBRANES ESOCAP AG (CH) 2025-12-04 US claimed
US-20250188088-A1 COMPOUND AND USE THEREOF ONQUALITY PHARMACEUTICALS CHINA LTD. (CN) 2025-06-12 US claimed
CN-119325375-A Drug delivery system comprising an anti-inflammatory agent or a salt thereof for application to the esophageal mucosa 伊斯凯普公司 2025-01-17 CN claimed
EP-4484429-A1 COMPOUND AND USE THEREOF OnQuality Pharmaceuticals China Ltd. (CN) 2025-01-01 EP claimed
CN-118715226-A Compounds and uses thereof 上海岸阔医药科技有限公司 2024-09-27 CN claimed
US-20240139327-A1 PRODRUG COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF MINGHUI PHARMACEUTICAL (HANGZHOU) LIMITED (CN) 2024-05-02 US claimed
EP-4293020-A1 PRODRUG COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Minghui Pharmaceutical (Hangzhou) Limited (CN) 2023-12-20 EP claimed
WO-2023237425-A1 DRUG DELIVERY SYSTEM COMPRISING AN ANTI-INFLAMMATORY AGENT OR A SALT THEREOF FOR THE APPLICATION TO ESOPHAGEAL MUCOUS MEMBRANES ESOCAP AG (CH) 2023-12-14 WO claimed
US-20230293503-A1 USE OF BERBERINE ANALOG AND JAK INHIBITOR IN TREATMENT OF INFLAMMATORY DISEASES OF GASTROINTESTINAL TRACT ENNOVABIO (ZHEJIANG) PHARMACEUTICALS CO., LTD. (CN) 2023-09-21 US claimed
US-20230271982-A1 CODRUG THAT DISINTEGRATES IN INTESTINE, PREPARATION THEREFOR, AND USE THEREOF SHANGHAI ENNOVABIO PHARMACEUTICALS CO., LTD. (CN) 2023-08-31 US claimed
WO-2023155905-A1 COMPOUND AND USE THEREOF 上海岸阔医药科技有限公司 2023-08-24 WO claimed
US-20230233158-A1 COMPUTERIZED DECISION SUPPORT TOOL AND MEDICAL DEVICE FOR SCRATCH DETECTION AND FLARE PREDICTION PFIZER INC. (US) 2023-07-27 US claimed
CN-116249533-A Intestinal tract cracking type co-drug and preparation and application thereof 轶诺(浙江)药业有限公司 2023-06-09 CN claimed
EP-4186900-A1 CODRUG THAT DISINTEGRATES IN INTESTINE, PREPARATION THEREFOR, AND USE THEREOF Ennovabio (Zhejiang) Pharmaceuticals Co., Ltd. (CN) 2023-05-31 EP claimed
EP-4167838-A1 COMPUTERIZED DECISION SUPPORT TOOL AND MEDICAL DEVICE FOR SCRATCH DETECTION AND FLARE PREDICTION Pfizer Inc. (US) 2023-04-26 EP claimed
CN-116018653-A Computerized decision support tool and medical device for scratch detection and seizure prediction 辉瑞公司 2023-04-25 CN claimed
WO-2022171140-A1 PRODRUG COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 明慧医药(杭州)有限公司 2022-08-18 WO claimed
CN-114907353-A Prodrug compound and preparation method and application thereof 明慧医药(杭州)有限公司 2022-08-16 CN claimed
EP-4167838-B1 COMPUTERIZED DECISION SUPPORT TOOL AND MEDICAL DEVICE FOR SCRATCH DETECTION AND FLARE PREDICTION PFIZER (US) 2026-05-20 EP disclosed
US-12617805-B2 Codrug that disintegrates in intestine, preparation therefor, and use thereof ENNOVABIO (ZHEJIANG) PHARMACEUTICALS CO., LTD. (CN) 2026-05-05 US disclosed
US-12594339-B2 Lipid prodrugs of JAK inhibitors and uses thereof SEAPORT THERAPEUTICS, INC. (US) 2026-04-07 US disclosed
US-20260021096-A1 TREATMENT OF HIDRADENITIS SUPPURATIVA USING JAK INHIBITORS INCYTE CORPORATION (US) 2026-01-22 US disclosed
EP-4662319-A2 PERSONALIZED CRISPR PROFILING FOR CANCER Integrate Bioscience LLC (US) 2025-12-17 EP disclosed
US-12498382-B2 Biomarkers for vitiligo INCYTE CORPORATION (US) 2025-12-16 US disclosed
US-20250367113-A1 DRUG DELIVERY SYSTEM COMPRISING AN ANTI-INFLAMMATORY AGENT OR A SALT THEREOF FOR THE APPLICATION TO ESOPHAGEAL MUCOUS MEMBRANES ESOCAP AG (CH) 2025-12-04 US disclosed
WO-2025226637-A1 COMBINATION THERAPY WITH AN ANTI-COLONY STIMULATING FACTOR 1 RECEPTOR ANTIBODY AND A JAK INHIBITOR INCYTE CORPORATION (US) 2025-10-30 WO disclosed
US-20250325664-A1 COMBINATION THERAPY WITH AN ANTI-COLONY STIMULATING FACTOR 1 RECEPTOR ANTIBODY AND A JAK INHIBITOR INCYTE CORP (US) 2025-10-23 US disclosed
EP-4590700-A1 TREATING SKIN IRRITATION FROM APPLICATION OF AN ALTERNATING ELECTRIC FIELD Novocure GmbH (CH) 2025-07-30 EP disclosed
US-12360120-B2 Biomarkers for graft-versus-host disease INCYTE CORPORATION (US) 2025-07-15 US disclosed
EP-4570321-A2 JAK INHIBITOR WITH A VITAMIN D ANALOG FOR TREATMENT OF SKIN DISEASES Incyte Corporation (US) 2025-06-18 EP disclosed
US-20250188088-A1 COMPOUND AND USE THEREOF ONQUALITY PHARMACEUTICALS CHINA LTD. (CN) 2025-06-12 US disclosed
WO-2025121754-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING SKIN DISEASES COMPRISING JANUS KINASE INHIBITOR 장병모 2025-06-12 WO disclosed
US-12280054-B2 Treatment of hidradenitis suppurativa using JAK inhibitors INCYTE CORPORATION (US) 2025-04-22 US disclosed
EP-4255442-B1 JAK INHIBITOR WITH A VITAMIN D ANALOG FOR TREATMENT OF SKIN DISEASES INCYTE CORP (US) 2025-03-19 EP disclosed
US-20250049817-A1 JAK INHIBITOR WITH A VITAMIN D ANALOG FOR TREATMENT OF SKIN DISEASES INCYTE CORP (US) 2025-02-13 US disclosed
US-12203942-B2 Biomarkers for graft-versus-host disease INCYTE CORPORATION (US) 2025-01-21 US disclosed
CN-119325375-A Drug delivery system comprising an anti-inflammatory agent or a salt thereof for application to the esophageal mucosa 伊斯凯普公司 2025-01-17 CN disclosed
EP-4484429-A1 COMPOUND AND USE THEREOF OnQuality Pharmaceuticals China Ltd. (CN) 2025-01-01 EP disclosed
US-20240390378-A1 USE OF JAK1 INHIBITORS FOR THE TREATMENT OF CUTANEOUS LUPUS ERYTHEMATOSUS AND LICHEN PLANUS (LP) INCYTE CORPORATION 2024-11-28 US disclosed
CN-118715226-A Compounds and uses thereof 上海岸阔医药科技有限公司 2024-09-27 CN disclosed
US-12099068-B2 Biomarkers for graft-versus-host disease INCYTE CORPORATION (US) 2024-09-24 US disclosed
EP-4424328-A2 TREATMENT OF HIDRADENITIS SUPPURATIVA USING JAK INHIBITORS Incyte Corporation (US) 2024-09-04 EP disclosed
CN-113166177-B Boron-containing PDE4 inhibitors 辉瑞公司 2024-09-03 CN disclosed
WO-2024168301-A2 PERSONALIZED CRISPR PROFILING FOR CANCER FUNCTION ONCOLOGY, INC. (US) 2024-08-15 WO disclosed
US-12005067-B2 JAK inhibitor with a vitamin D analog for treatment of skin diseases INCYTE CORPORATION (US) 2024-06-11 US disclosed
US-11992490-B2 Use of JAK1 inhibitors for the treatment of cutaneous lupus erythematosus and Lichen planus (LP) INCYTE CORPORATION (US) 2024-05-28 US disclosed
US-20240139327-A1 PRODRUG COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF MINGHUI PHARMACEUTICAL (HANGZHOU) LIMITED (CN) 2024-05-02 US disclosed
US-20240132477-A1 Benzimidazole Derivatives and Their Use As Inhibitors of ITK For The Treatment of Skin Disease PFIZER INC. (US) 2024-04-25 US disclosed
US-20240124439-A1 Pyrido[2,3-D]Imidazole Derivatives and Their Use As Inhibitors of ITK for the Treatment of Skin Disease PFIZER INC. (US) 2024-04-18 US disclosed
CN-115361974-B Use of berberine analogues and JAK inhibitors in the treatment of inflammatory diseases of the gastrointestinal tract 轶诺(浙江)药业有限公司 2024-04-16 CN disclosed
WO-2024062457-A1 TREATING SKIN IRRITATION FROM APPLICATION OF AN ALTERNATING ELECTRIC FIELD NOVOCURE GMBH (CH) 2024-03-28 WO disclosed
US-20240101661-A1 TREATING SKIN IRRITATION FROM APPLICATION OF AN ALTERNATING ELECTRIC FIELD NOVOCURE GMBH (CH) 2024-03-28 US disclosed
EP-4293020-A1 PRODRUG COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Minghui Pharmaceutical (Hangzhou) Limited (CN) 2023-12-20 EP disclosed
WO-2023237425-A1 DRUG DELIVERY SYSTEM COMPRISING AN ANTI-INFLAMMATORY AGENT OR A SALT THEREOF FOR THE APPLICATION TO ESOPHAGEAL MUCOUS MEMBRANES ESOCAP AG (CH) 2023-12-14 WO disclosed
EP-3861001-B1 BORON CONTAINING PDE4 INHIBITORS PFIZER (US) 2023-12-13 EP disclosed
CN-117157080-A JAK inhibitors containing vitamin D analogues for the treatment of skin disorders 因赛特公司 2023-12-01 CN disclosed
EP-4263526-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS INHIBITORS OF ITK FOR THE TREATMENT OF SKIN DISEASE Pfizer Inc. (US) 2023-10-25 EP disclosed
EP-4263538-A1 PYRIDO[2,3-D]IMIDAZOLE DERIVATIVES AND THEIR USE AS INHIBITORS OF ITK FOR THE TEATMENT OF SKIN DISEASE Pfizer Inc. (US) 2023-10-25 EP disclosed
EP-4255442-A1 JAK INHIBITOR WITH A VITAMIN D ANALOG FOR TREATMENT OF SKIN DISEASES Incyte Corporation (US) 2023-10-11 EP disclosed
US-20230293503-A1 USE OF BERBERINE ANALOG AND JAK INHIBITOR IN TREATMENT OF INFLAMMATORY DISEASES OF GASTROINTESTINAL TRACT ENNOVABIO (ZHEJIANG) PHARMACEUTICALS CO., LTD. (CN) 2023-09-21 US disclosed
US-20230280220-A1 Benzimidazole Derivative Compounds and Uses Thereof PFIZER INC. (US) 2023-09-07 US disclosed
US-20230271982-A1 CODRUG THAT DISINTEGRATES IN INTESTINE, PREPARATION THEREFOR, AND USE THEREOF SHANGHAI ENNOVABIO PHARMACEUTICALS CO., LTD. (CN) 2023-08-31 US disclosed
WO-2023155905-A1 COMPOUND AND USE THEREOF 上海岸阔医药科技有限公司 2023-08-24 WO disclosed
US-20230233158-A1 COMPUTERIZED DECISION SUPPORT TOOL AND MEDICAL DEVICE FOR SCRATCH DETECTION AND FLARE PREDICTION PFIZER INC. (US) 2023-07-27 US disclosed
US-20230220478-A1 BIOMARKERS FOR VITILIGO INCYTE CORPORATION 2023-07-13 US disclosed
CN-116249533-A Intestinal tract cracking type co-drug and preparation and application thereof 轶诺(浙江)药业有限公司 2023-06-09 CN disclosed
EP-4186900-A1 CODRUG THAT DISINTEGRATES IN INTESTINE, PREPARATION THEREFOR, AND USE THEREOF Ennovabio (Zhejiang) Pharmaceuticals Co., Ltd. (CN) 2023-05-31 EP disclosed
US-11661419-B2 Benzimidazole derivative compounds and uses thereof PFIZER INC. (US) 2023-05-30 US disclosed
US-20230148402-A1 Boron Containing PDE4 Inhibitors PFIZER INC. (US) 2023-05-11 US disclosed
EP-4167838-A1 COMPUTERIZED DECISION SUPPORT TOOL AND MEDICAL DEVICE FOR SCRATCH DETECTION AND FLARE PREDICTION Pfizer Inc. (US) 2023-04-26 EP disclosed
CN-116018653-A Computerized decision support tool and medical device for scratch detection and seizure prediction 辉瑞公司 2023-04-25 CN disclosed
US-11624751-B2 Biomarkers for vitiligo INCYTE CORPORATION (US) 2023-04-11 US disclosed
CN-112533606-B Application of JAK kinase inhibitor and EGFR inhibitor in preparation of medicines for treating tumor diseases 江苏恒瑞医药股份有限公司 2023-04-04 CN disclosed
US-11584961-B2 Biomarkers for inflammatory skin disease INCYTE CORPORATION (US) 2023-02-21 US disclosed
US-20230027606-A1 BIOMARKERS FOR GRAFT-VERSUS-HOST DISEASE INCYTE CORPORATION 2023-01-26 US disclosed
US-11559538-B2 Substituted 1,2-oxaborolan-2-ols as PDE4 inhibitors PFIZER INC. (US) 2023-01-24 US disclosed
EP-4077316-A1 BENZIMIDAZOLE DERIVATIVES Pfizer Inc. (US) 2022-10-26 EP disclosed
WO-2022171140-A1 PRODRUG COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 明慧医药(杭州)有限公司 2022-08-18 WO disclosed
CN-114907353-A Prodrug compound and preparation method and application thereof 明慧医药(杭州)有限公司 2022-08-16 CN disclosed
CN-111094314-B Prodrug containing glucuronide derivative JAK inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2022-08-12 CN disclosed
US-20220241286-A1 TREATMENT OF HIDRADENITIS SUPPURATIVA USING JAK INHIBITORS INCYTE CORPORATION 2022-08-04 US disclosed
US-20220202834-A1 JAK INHIBITOR WITH A VITAMIN D ANALOG FOR TREATMENT OF SKIN DISEASES INCYTE CORPORATION 2022-06-30 US disclosed
US-11372003-B2 Biomarkers for graft-versus-host disease INCYTE CORPORATION (US) 2022-06-28 US disclosed
WO-2022130175-A1 PYRIDO[2,3-D]IMIDAZOLE DERIVATIVES AND THEIR USE AS INHIBITORS OF ITK FOR THE TEATMENT OF SKIN DISEASE PFIZER INC. (US) 2022-06-23 WO disclosed
WO-2022130171-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS INHIBITORS OF ITK FOR THE TREATMENT OF SKIN DISEASE PFIZER INC. (US) 2022-06-23 WO disclosed
WO-2022120131-A1 JAK INHIBITOR WITH A VITAMIN D ANALOG FOR TREATMENT OF SKIN DISEASES INCYTE CORPORATION (US) 2022-06-09 WO disclosed
US-20220125933-A1 LIPID PRODRUGS OF JAK INHIBITORS AND USES THEREOF SEAPORT THERAPEUTICS, INC. 2022-04-28 US disclosed
US-11304949-B2 Treatment of hidradenitis suppurativa using JAK inhibitors INCYTE CORPORATION (US) 2022-04-19 US disclosed
EP-3941474-A2 BIOMARKERS FOR VITILIGO Incyte Corporation (US) 2022-01-26 EP disclosed
EP-3941474-A2 BIOMARKERS FOR VITILIGO Incyte Corporation (US) 2022-01-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (29 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11559538-B2 Substituted 1,2-oxaborolan-2-ols as PDE4 inhibitors PDE4B, PDE4A, PDE3B JAK1 2263/4885JAK3 2865/4885JAK2 2446/4885
US-12005067-B2 JAK inhibitor with a vitamin D analog for treatment of skin diseases JAK3, IL23R, JAK1 JAK1 3/4885JAK3 1/4885JAK2 5/4885
US-11372003-B2 Biomarkers for graft-versus-host disease CD74, HLA-DRB1, TSG101 JAK1 5/4885JAK3 4/4885JAK2 26/4885
US-20220125933-A1 LIPID PRODRUGS OF JAK INHIBITORS AND USES THEREOF JAK1, JAK2, JAK3 JAK1 1/4885JAK3 3/4885JAK2 2/4885
US-11304949-B2 Treatment of hidradenitis suppurativa using JAK inhibitors JAK1, JAK2, JAK3 JAK1 1/4885JAK3 3/4885JAK2 2/4885
US-20240132477-A1 Benzimidazole Derivatives and Their Use As Inhibitors of ITK For The Treatment of Skin Disease ITK, BLK, BCKDK JAK1 59/4885JAK3 125/4885JAK2 208/4885
US-20240390378-A1 USE OF JAK1 INHIBITORS FOR THE TREATMENT OF CUTANEOUS LUPUS ERYTHEMATOSUS AND LICHEN PLANUS (LP) JAK1, JAK3, JAK2 JAK1 1/4885JAK3 2/4885JAK2 3/4885
US-12360120-B2 Biomarkers for graft-versus-host disease CD74, HLA-DRB1, TSG101 JAK1 7/4885JAK3 6/4885JAK2 38/4885
US-12498382-B2 Biomarkers for vitiligo TSG101, JAK3, IFNG JAK1 5/4885JAK3 2/4885JAK2 13/4885
US-20240139327-A1 PRODRUG COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF CYP51A1, CYP4F11, NOTUM JAK1 3194/4885JAK3 4246/4885JAK2 4085/4885
US-20260021096-A1 TREATMENT OF HIDRADENITIS SUPPURATIVA USING JAK INHIBITORS JAK1, JAK2, JAK3 JAK1 1/4885JAK3 3/4885JAK2 2/4885
US-20250325664-A1 COMBINATION THERAPY WITH AN ANTI-COLONY STIMULATING FACTOR 1 RECEPTOR ANTIBODY AND A JAK INHIBITOR JAK1, CSF3R, JAK3 JAK1 1/4885JAK3 3/4885JAK2 5/4885
US-20220241286-A1 TREATMENT OF HIDRADENITIS SUPPURATIVA USING JAK INHIBITORS JAK1, JAK2, JAK3 JAK1 1/4885JAK3 3/4885JAK2 2/4885
US-20250049817-A1 JAK INHIBITOR WITH A VITAMIN D ANALOG FOR TREATMENT OF SKIN DISEASES JAK3, IL23R, JAK1 JAK1 3/4885JAK3 1/4885JAK2 5/4885
US-12099068-B2 Biomarkers for graft-versus-host disease CD74, HLA-DRB1, TSG101 JAK1 5/4885JAK3 4/4885JAK2 26/4885
US-20230148402-A1 Boron Containing PDE4 Inhibitors PDE4B, PDE4A, PDE3B JAK1 1657/4885JAK3 1949/4885JAK2 1684/4885
US-20230293503-A1 USE OF BERBERINE ANALOG AND JAK INHIBITOR IN TREATMENT OF INFLAMMATORY DISEASES OF GASTROINTESTINAL TRACT JAK1, JAK2, JAK3 JAK1 1/4885JAK3 3/4885JAK2 2/4885
US-12617805-B2 Codrug that disintegrates in intestine, preparation therefor, and use thereof IRAK4, JAK1, VIP JAK1 2/4885JAK3 14/4885JAK2 26/4885
US-11624751-B2 Biomarkers for vitiligo TSG101, JAK3, IFNG JAK1 5/4885JAK3 2/4885JAK2 13/4885
US-20220202834-A1 JAK INHIBITOR WITH A VITAMIN D ANALOG FOR TREATMENT OF SKIN DISEASES JAK3, IL23R, JAK1 JAK1 3/4885JAK3 1/4885JAK2 5/4885
US-20240124439-A1 Pyrido[2,3-D]Imidazole Derivatives and Their Use As Inhibitors of ITK for the Treatment of Skin Disease ITK, PDXK, HRH4 JAK1 162/4885JAK3 134/4885JAK2 660/4885
US-11661419-B2 Benzimidazole derivative compounds and uses thereof ITK, HRH4, BLK JAK1 93/4885JAK3 189/4885JAK2 173/4885
US-12594339-B2 Lipid prodrugs of JAK inhibitors and uses thereof JAK1, JAK3, JAK2 JAK1 1/4885JAK3 2/4885JAK2 3/4885
US-20230271982-A1 CODRUG THAT DISINTEGRATES IN INTESTINE, PREPARATION THEREFOR, AND USE THEREOF VIP, SI, PDCD5 JAK1 2922/4885JAK3 3340/4885JAK2 4173/4885
US-12203942-B2 Biomarkers for graft-versus-host disease CD74, HLA-DRB1, TSG101 JAK1 7/4885JAK3 6/4885JAK2 38/4885
US-12280054-B2 Treatment of hidradenitis suppurativa using JAK inhibitors JAK1, JAK2, JAK3 JAK1 1/4885JAK3 3/4885JAK2 2/4885
US-20250188088-A1 COMPOUND AND USE THEREOF CYP17A1, CYP11B2, CYP21A2 JAK1 3705/4885JAK3 4037/4885JAK2 1497/4885
US-11992490-B2 Use of JAK1 inhibitors for the treatment of cutaneous lupus erythematosus and Lichen planus (LP) JAK1, JAK3, JAK2 JAK1 1/4885JAK3 2/4885JAK2 3/4885
US-20230027606-A1 BIOMARKERS FOR GRAFT-VERSUS-HOST DISEASE CD74, HLA-DRB1, TSG101 JAK1 5/4885JAK3 4/4885JAK2 26/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.