Gsk-650394

Gsk-650394

SCHEMBL29368746

O=C(O)c1ccc(-c2c[nH]c3ncc(-c4ccccc4)cc23)cc1C1CCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 17/20 1.00
CAMKK1 Q8N5S9 4/20 1.00
SGK1 O00141 3/20 1.00
AURKA O14965 1/20 1.00
SGK3 Q96BR1 1/20 1.00
SGK2 Q9HBY8 1/20 1.00
AXL P30530 4/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gsk-650394 SCHEMBL30753539 1.00 CAMKK2 (1.00) CAMKK2CAMKK1SGK1AURKASGK3
Gsk-650394 SCHEMBL3767908 1.00 CAMKK2 (1.00) CAMKK2CAMKK1SGK1AURKASGK3
SCHEMBL3767383 0.81 CAMKK2 (1.00) CAMKK2CAMKK1SGK1AURKASGK3
SCHEMBL3768084 0.79 CAMKK2 (1.00) CAMKK2CAMKK1SGK1AURKASGK3
SCHEMBL3767167 0.79 CAMKK2 (0.76) CAMKK2CAMKK1SGK1AURKASGK3
SCHEMBL3762417 0.78 CAMKK2 (0.74) CAMKK2CAMKK1SGK1AURKASGK3
SCHEMBL3764354 0.78 CAMKK2 (0.82) CAMKK2CAMKK1SGK1AURKASGK3
SCHEMBL3766865 0.78 CAMKK2 (1.00) CAMKK2CAMKK1SGK1AURKASGK3
SCHEMBL3774587 0.77 AXL (1.00) CAMKK2SGK1AURKASGK2AXL
SCHEMBL3759420 0.77 AXL (1.00) CAMKK2SGK1AURKASGK2AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119818491-A Application of SGK1 inhibitor in preparation of medicine for treating endometriosis 中国福利会国际和平妇幼保健院 2025-04-15 CN claimed
US-20230364086-A1 COMBINATION THERAPIES WITH EHMT2 INHIBITORS Epizyme, Inc. 2023-11-16 US claimed
US-20230218634-A1 METHODS OF TREATING CASTRATION-RESISTANT PROSTATE CANCER WITH GLUCOCORTICOID RECEPTOR ANTAGONISTS AND ANTI-ANDROGEN RECEPTOR THERAPY AND ANTI-ANDROGEN RECEPTOR THERAPY UNIVERSITY OF CHICAGO (US) 2023-07-13 US claimed
US-11564932-B2 Methods of treating castration-resistant prostate cancer with glucocorticoid receptor antagonists and anti-androgen receptor therapy THE UNIVERSITY OF CHICAGO (US) 2023-01-31 US claimed
US-20220259654-A1 COMPOSITIONS AND METHODS FOR XI CHROMOSOME REACTIVATION UNIVERSITY OF MASSACHUSETTS (US) 2022-08-18 US claimed
US-20260024617-A1 METHODS AND SYSTEMS FOR PERSONALIZED THERAPIES SCIPHER MEDICINE CORP (US) 2026-01-22 US disclosed
US-12303549-B2 Methods of treating or inhibiting onset of Huntington's disease UNIVERSITY OF ROCHESTER (US) 2025-05-20 US disclosed
US-12295955-B2 TTP phosphorylation for the identification of personalized medicines KING FAISAL SPECIALIST HOSPITAL & RESEARCH CENTRE (SA) 2025-05-13 US disclosed
CN-119950724-A Application of SGK1 as marker in tumor immunotherapy 北京大学 2025-05-09 CN disclosed
CN-119818491-A Application of SGK1 inhibitor in preparation of medicine for treating endometriosis 中国福利会国际和平妇幼保健院 2025-04-15 CN disclosed
CN-119818491-A Application of SGK1 inhibitor in preparation of medicine for treating endometriosis 中国福利会国际和平妇幼保健院 2025-04-15 CN disclosed
EP-4529477-A1 POROUS EXPANDING BIOCOMPATIBLE SCAFFOLDS Danmarks Tekniske Universitet (DK) 2025-04-02 EP disclosed
US-20220339285-A1 DISSACHARIDE FORMULATIONS FOR CONTROLLED DRUG RELEASE TECHNICAL UNIVERSITY OF DENMARK (DK) 2022-10-27 US disclosed
CN-115006536-A Application of Sgk1 as target in preparation of medicine for inhibiting gluconeogenesis 上海交通大学医学院附属瑞金医院 2022-09-06 CN disclosed
US-20220259654-A1 COMPOSITIONS AND METHODS FOR XI CHROMOSOME REACTIVATION UNIVERSITY OF MASSACHUSETTS (US) 2022-08-18 US disclosed
US-20220244263-A1 METHODS FOR TREATING SMALL CELL NEUROENDOCRINE AND RELATED CANCERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-08-04 US disclosed
US-11389432-B2 Methods of treating cancer comprising administration of a glucocorticoid receptor modulator and a cancer chemotherapy agent CORCEPT THERAPEUTICS INCORPORATED (US) 2022-07-19 US disclosed
EP-3982922-A1 DISSACHARIDE FORMULATIONS FOR CONTROLLED DRUG RELEASE Technical University of Denmark (DK) 2022-04-20 EP disclosed
US-20220062378-A1 METHODS OF TREATING OR INHIBITING ONSET OF HUNTINGTON'S DISEASE UNIVERSITY OF COPENHAGEN (DK) 2022-03-03 US disclosed
US-11234971-B2 Methods of treating cancer comprising administration of a glucocorticoid receptor modulator and a cancer chemotherapy agent CORCEPT THERAPEUTICS INCORPORATED (US) 2022-02-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230364086-A1 COMBINATION THERAPIES WITH EHMT2 INHIBITORS EHMT2, BHMT, SHMT2 CAMKK2 1862/4885CAMKK1 2729/4885SGK1 1590/4885
US-11389432-B2 Methods of treating cancer comprising administration of a glucocorticoid receptor modulator and a cancer chemotherapy agent NR3C1, GRK2, GRK3 CAMKK2 228/4885CAMKK1 307/4885SGK1 4/4885
US-11234971-B2 Methods of treating cancer comprising administration of a glucocorticoid receptor modulator and a cancer chemotherapy agent NR3C1, GRK4, GRK5 CAMKK2 1027/4885CAMKK1 1449/4885SGK1 60/4885
US-20260024617-A1 METHODS AND SYSTEMS FOR PERSONALIZED THERAPIES SET, SSB, CNKSR1 CAMKK2 1213/4885CAMKK1 1630/4885SGK1 3969/4885
US-20220339285-A1 DISSACHARIDE FORMULATIONS FOR CONTROLLED DRUG RELEASE LIPA, LIPE, CEL CAMKK2 1273/4885CAMKK1 1174/4885SGK1 1613/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.