Flupirtine

Flupirtine

SCHEMBL29400613

CCOC(=O)Nc1ccc(NCc2ccc(F)cc2)nc1N

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 9/20 1.00
KCNQ3 O43525 7/20 1.00
CYP1A2 P05177 2/20 1.00
CYP2C9 P11712 2/20 1.00
CYP2C19 P33261 2/20 1.00
ABCB11 O95342 1/20 1.00
ESR1 P03372 1/20 1.00
CYP3A4 P08684 1/20 1.00
HTR1A P08908 1/20 1.00
ADRA2A P08913 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
CYP2D6 P10635 1/20 1.00
ALOX15 P16050 1/20 1.00
NFKB1 P19838 1/20 1.00
TBXA2R P21731 1/20 1.00
MAPK1 P28482 1/20 1.00
CASP1 P29466 1/20 1.00
SHMT2 P34897 1/20 1.00
PTGS2 P35354 1/20 1.00
OPRK1 P41145 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flupirtine SCHEMBL3896230 1.00 KCNQ2 (1.00) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL15357226 1.00 KCNQ2 (1.00) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL25009 1.00 KCNQ2 (1.00) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL505847 0.99 KCNQ2 (0.98) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL505535 0.99 KCNQ2 (0.98) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL28262990 0.99 KCNQ2 (0.98) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL505446 0.98 KCNQ2 (0.96) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL505680 0.98 KCNQ2 (0.96) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL1649863 0.98 KCNQ2 (0.96) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19
Flupirtine SCHEMBL505608 0.97 KCNQ2 (0.94) KCNQ2KCNQ3CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 118 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
WO-2025104452-A1 COMPOUNDS FOR USE IN TREATMENT MITORX THERAPEUTICS LTD (GB) 2025-05-22 WO claimed
WO-2024015527-A1 THERAPEUTIC COMBINATIONS OF DRUGS, COMPANION DIAGNOSTICS AND METHODS FOR DOSAGING AND USING THEM BAYESIAN BIOTECH, LLC (US) 2024-01-18 WO claimed
EP-3682872-B1 LIQUISOFT CAPSULES PATHEON SOFTGELS INC (US) 2024-01-03 EP claimed
EP-3380121-B1 ACTRII ANTAGONIST FOR USE IN TREATING EYE DISORDERS ACCELERON PHARMA INC (US) 2023-12-20 EP claimed
US-12605470-B2 Nanodroplet with layer-by-layer assembly ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2026-04-21 US disclosed
US-20260083770-A1 RNA COMPLEXES AND NANOSTRUCTURES FOR TREATMENT OF CANCER METASTASIS OHIO STATE INNOVATION FOUNDATION (US) 2026-03-26 US disclosed
EP-4714496-A2 TREATMENT OF NEURONAL CEROID LIPOFUSCINOSIS OrfoNeuro ApS (DK) 2026-03-25 EP disclosed
US-20260077027-A1 PEPTIDE AND NUCLEIC ACID METHODS TO MODULATE DELIVERY OF NUCLEIC ACID STRUCTURES, POLYPEPTIDES, AND THEIR CARGOES OHIO STATE INNOVATION FOUNDATION (US) 2026-03-19 US disclosed
US-12577282-B2 Galectin-1/ galectin-3 chimeras and multivalent proteins UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2026-03-17 US disclosed
EP-4706683-A2 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2026-03-11 EP disclosed
US-20260053906-A1 DNA ORIGAMI VACCINES OHIO STATE INNOVATION FOUNDATION (US) 2026-02-26 US disclosed
US-11369593-B2 Functionalized pyridine carbamates with enhanced neuroprotective activity TEXAS TECH UNIVERSITY SYSTEM (US) 2022-06-28 US disclosed
US-20220175804-A1 aPKC INHIBITORS AND METHODS OF TREATING A NEURODEGENERATIVE DISEASE OR DISORDER THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2022-06-09 US disclosed
US-11324855-B2 Cell-free combination, hydrogel-like material or hydrogel and use of same TETEC TISSUE ENGINEERING TECHNOLOGIES AG (DE) 2022-05-10 US disclosed
WO-2022076932-A1 COMPOSITIONS AND METHODS OF TREATING A PI3K MEDIATED DISEASE VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 2022-04-14 WO disclosed
US-20220106580-A1 TARGETED CHONDROITINASE ABC FUSION PROTEINS AND COMPLEXES THEREOF UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2022-04-07 US disclosed
US-20220098258-A1 GALECTIN-1/ GALECTIN-3 CHIMERAS AND MULTIVALENT PROTEINS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2022-03-31 US disclosed
WO-2022049149-A1 CHEWABLE FORMULATIONS ELANCO TIERGESUNDHEIT AG (CH) 2022-03-10 WO disclosed
US-20220054649-A1 ANTIBODY-DRUG CONJUGATES SPIREA LIMITED (GB) 2022-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12577282-B2 Galectin-1/ galectin-3 chimeras and multivalent proteins LGALS1, LGALS3BP, LGALS3 KCNQ2 4216/4885KCNQ3 3538/4885CYP1A2 4831/4885
US-20260053906-A1 DNA ORIGAMI VACCINES CD47, RBM26, TP53 KCNQ2 2568/4885KCNQ3 2364/4885CYP1A2 4867/4885
US-11369593-B2 Functionalized pyridine carbamates with enhanced neuroprotective activity BDNF, CHRNA5, CHRNA4 KCNQ2 783/4885KCNQ3 852/4885CYP1A2 1609/4885
US-20260083770-A1 RNA COMPLEXES AND NANOSTRUCTURES FOR TREATMENT OF CANCER METASTASIS RNMT, NSUN2, FBL KCNQ2 4325/4885KCNQ3 4239/4885CYP1A2 4679/4885
US-20220054649-A1 ANTIBODY-DRUG CONJUGATES CD44, CD47, FCGR3B KCNQ2 3807/4885KCNQ3 3774/4885CYP1A2 2004/4885
US-20260077027-A1 PEPTIDE AND NUCLEIC ACID METHODS TO MODULATE DELIVERY OF NUCLEIC ACID STRUCTURES, POLYPEPTIDES, AND THEIR CARGOES MICA, PDCD1LG2, TLR9 KCNQ2 4279/4885KCNQ3 4094/4885CYP1A2 4882/4885
US-12605470-B2 Nanodroplet with layer-by-layer assembly FLNB, FLNA, DAGLB KCNQ2 3598/4885KCNQ3 3240/4885CYP1A2 4594/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.