Nicomorphine

Nicomorphine

SCHEMBL29408441

CN1CC[C@]23c4c5ccc(OC(=O)c6cccnc6)c4O[C@H]2[C@@H](OC(=O)c2cccnc2)C=C[C@H]3[C@H]1C5

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 10/20 0.69
OPRM1 P35372 12/20 0.60
OPRK1 P41145 10/20 0.60
ADRB1 P08588 1/20 0.53
PDE4D Q08499 1/20 0.53
PDE3A Q14432 1/20 0.53
MRGPRX2 Q96LB1 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nicomorphine SCHEMBL680036 1.00 OPRD1 (0.69) OPRD1OPRM1OPRK1ADRB1PDE4D
Nicomorphine SCHEMBL26237 1.00 OPRD1 (0.69) OPRD1OPRM1OPRK1ADRB1PDE4D
Nicomorphine SCHEMBL29349768 1.00 OPRD1 (0.69) OPRD1OPRM1OPRK1ADRB1PDE4D
Nicomorphine SCHEMBL1649977 0.99 OPRD1 (0.68) OPRD1OPRM1OPRK1ADRB1PDE4D
Nicomorphine SCHEMBL395672 0.99 OPRD1 (0.68) OPRD1OPRM1OPRK1ADRB1PDE4D
Nicocodine SCHEMBL1023092 0.94 OPRM1 (0.69) OPRD1OPRM1OPRK1ADRB1PDE4D
Nicocodine SCHEMBL159020 0.94 OPRM1 (0.69) OPRD1OPRM1OPRK1ADRB1PDE4D
Nicocodine SCHEMBL29531263 0.94 OPRM1 (0.69) OPRD1OPRM1OPRK1ADRB1PDE4D
SCHEMBL27496008 0.91 OPRD1 (0.66) OPRD1OPRM1OPRK1ADRB1PDE4D
SCHEMBL1556900 0.91 OPRD1 (0.82) OPRD1OPRM1OPRK1ADRB1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3682872-B1 LIQUISOFT CAPSULES PATHEON SOFTGELS INC (US) 2024-01-03 EP claimed
EP-3064199-B1 ABUSE-DETERRENT TRANSDERMAL FORMULATIONS OF OPIATE AGONISTS AND AGONIST-ANTAGONISTS BUZZZ PHARMACEUTICALS LTD (IE) 2023-12-20 EP claimed
EP-3405179-B1 CONTROL OF THE RELEASE OF WATER FROM A SOLID COMPOSITION CONTAINING WATER LTS LOHMANN THERAPIE SYSTEME AG (DE) 2023-08-09 EP claimed
EP-3528804-B1 CHEWING GUM COMPOSITION COMPRISING CANNABINOIDS AND OPIOID AGONISTS AND/OR ANTAGONISTS APIRX PHARMACEUTICAL USA LLC (US) 2023-07-26 EP claimed
EP-3313407-B1 TREATMENT AND MANAGEMENT OF AUGMENTATION IN RESTLESS LEGS SYNDROME UNIV EAST CAROLINA (US) 2023-07-19 EP claimed
EP-3385252-B1 CANNABINOID RECEPTOR MODULATORS ARENA PHARM INC (US) 2022-09-21 EP claimed
EP-3291676-B1 MITRAGYNINE ANALOGS AND USES THEREOF MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-08-17 EP claimed
CN-114601834-A Use of mitochondrial fission inhibitors and combinations comprising the same 复旦大学 2022-06-10 CN claimed
CN-109553565-B Two new alkaloids, preparation method thereof and application thereof in preparation of MRSA-resistant antibacterial agent 华南农业大学 2022-04-05 CN claimed
CN-117772131-A Clay mineral-based carbon-silicon oxide nanocomposite and preparation method and application thereof 中国科学院广州地球化学研究所 2024-03-29 CN disclosed
EP-3405179-B1 CONTROL OF THE RELEASE OF WATER FROM A SOLID COMPOSITION CONTAINING WATER LTS LOHMANN THERAPIE SYSTEME AG (DE) 2023-08-09 EP disclosed
CN-116018131-A Fast orodispersible tablet with inner cavity 阿普雷奇亚制药有限责任公司 2023-04-25 CN disclosed
CN-115928318-A Preparation method of antibacterial and antiviral packaging material and packaging material using same 华南农业大学 2023-04-07 CN disclosed
CN-115942979-A MGLUR5 antagonist, marvorexant, for use in therapy to reduce opioid use 诺华股份有限公司 2023-04-07 CN disclosed
EP-1765303-B2 ORAL TABLET SAFEGUARDED AGAINST ABUSE GRUENENTHAL GMBH (DE) 2022-11-23 EP disclosed
CN-111132666-B Composition for delivering physiologically active ingredients to blood vessels 雷莫内克斯生物制药有限公司 2022-11-04 CN disclosed
CN-111632041-B Abuse resistant pharmaceutical composition 瑞克欧盖恩斯维尔有限责任公司 2022-10-04 CN disclosed
CN-115135323-A Pharmaceutical composition 深圳市药欣生物科技有限公司 2022-09-30 CN disclosed
CN-114601834-A Use of mitochondrial fission inhibitors and combinations comprising the same 复旦大学 2022-06-10 CN disclosed
CN-109689058-B Treatment and prevention of sleep disorders 普渡制药公司 2022-03-22 CN disclosed