Thiourea, N-(5-Bromo-2-Pyridinyl)-N'-(2-(2-Chloro-3-Ethoxy-6-Fluorophenyl)Ethyl)-

Thiourea, N-(5-Bromo-2-Pyridinyl)-N'-(2-(2-Chloro-3-Ethoxy-6-Fluorophenyl)Ethyl)-

SCHEMBL29422945

CCOc1ccc(F)c(CCNC(=S)Nc2ccc(Br)cn2)c1Cl

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
LTC4S Q16873 2/20 0.51
RAB9A P51151 5/20 0.41
MAPT P10636 5/20 0.41
NPC1 O15118 2/20 0.41
KMT2A Q03164 4/20 0.40
PKM P14618 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 1/20 0.40
MEN1 O00255 2/20 0.39
MAPK1 P28482 1/20 0.38
POLB P06746 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
GBA1 P04062 1/20 0.37
SSTR4 P31391 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiourea, N-(5-Bromo-2-Pyridinyl)-N'-(2-(2-Chloro-3-Ethoxy-6-Fluorophenyl)Ethyl)- SCHEMBL6906082 1.00 ALDH1A1 (0.52) ALDH1A1LTC4SRAB9AMAPTNPC1
SCHEMBL14439884 0.90 ALDH1A1 (0.54) ALDH1A1LTC4SRAB9AMAPTNPC1
SCHEMBL6905335 0.89 RAB9A (0.55) RAB9AMAPTNPC1KMT2ASMN1; SMN2
SCHEMBL6907153 0.89 ALDH1A1 (0.55) ALDH1A1LTC4SRAB9AMAPTNPC1
SCHEMBL2792582 0.86 ALDH1A1 (0.56) ALDH1A1LTC4SRAB9AMAPTNPC1
SCHEMBL29657174 0.83 ALDH1A1 (0.55) ALDH1A1LTC4SRAB9AMAPTNPC1
SCHEMBL6963627 0.83 ALDH1A1 (0.55) ALDH1A1LTC4SRAB9AMAPTNPC1
SCHEMBL14439886 0.81 ALDH1A1 (0.46) ALDH1A1LTC4SRAB9AMAPTNPC1
SCHEMBL6905477 0.80 ALDH1A1 (0.67) ALDH1A1LTC4SRAB9AMAPTNPC1
SCHEMBL14439885 0.78 LTC4S (0.61) ALDH1A1LTC4SRAB9AMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3565561-B1 PHOSPHAPLATIN COMPOUNDS AS THERAPEUTIC AGENTS FOR TREATMENT OF BONE BLOOD CANCERS PROMONTORY THERAPEUTICS INC (US) 2026-05-06 EP claimed
CN-118987015-A Application of antisense oligonucleotide in preparation of medicine for treating breast cancer 北京悦康科创医药科技股份有限公司 2024-11-22 CN claimed
EP-4460308-A2 COMPOSITIONS AND METHODS FOR TREATING CANCER OR PREVENTING, INHIBITING OR REDUCING RISK OF METASTASIS OF A CANCER Lixte Biotechnology, Inc. (US) 2024-11-13 EP claimed
US-20240317787-A1 ORGANIC ELECTROLUMINESCENT DEVICE Beijing Summer Sprout Technology Co., Ltd. (CN) 2024-09-26 US claimed
US-20240298520-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2024-09-05 US claimed
US-20240251654-A1 ORGANIC ELECTROLUMINESCENT DEVICE Beijing Summer Sprout Technology Co., Ltd. (CN) 2024-07-25 US claimed
EP-4003314-B1 FUNCTIONALIZED LONG-CHAIN HYDROCARBON MONO- AND DI-CARBOXYLIC ACIDS USEFUL FOR THE PREVENTION OR TREATMENT OF DISEASE ESPERVITA THERAPEUTICS INC (US) 2024-07-10 EP claimed
CN-118119386-A Functionalized carboxylic acids and their use for treating diseases 埃斯佩尔维塔治疗股份有限公司 2024-05-31 CN claimed
US-20240009212-A1 PHOSPHAPLATIN COMPOUNDS AS THERAPEUTIC AGENTS SELECTIVELY TARGETING HIGHLY GLYCOLYTIC TUMOR CELLS AND METHODS THEREOF PROMONTORY THERAPEUTICS INC. (US) 2024-01-11 US claimed
EP-4281058-A2 FUNCTIONALIZED LONG-CHAIN CARBOXYLIC ACIDS, AND THEIR USE FOR TREATMENT OF DISEASE Espervita Therapeutics, Inc. (US) 2023-11-29 EP claimed
EP-4232044-A1 PHOSPHAPLATIN COMPOUNDS AS THERAPEUTIC AGENTS SELECTIVELY TARGETING HIGHLY GLYCOLYTIC TUMOR CELLS AND METHODS THEREOF Promontory Therapeutics Inc. (US) 2023-08-30 EP claimed
WO-2023133371-A2 COMPOSITIONS AND METHODS FOR TREATING CANCER OR PREVENTING, INHIBITING OR REDUCING RISK OF METASTASIS OF A CANCER LIXTE BIOTECHNOLOGY, INC. (US) 2023-07-13 WO claimed
US-20230144846-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-05-11 US claimed
CN-115974931-A Organic electroluminescent material and device 环球展览公司 2023-04-18 CN claimed
US-20230111520-A1 FUNCTIONALIZED LONG-CHAIN HYDROCARBON MONO- AND DI-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF, AND THEIR USE FOR THE PREVENTION OR TREATMENT OF DISEASE ESPERVITA THERAPEUTICS, INC. 2023-04-13 US claimed
US-20230113853-A1 FUNCTIONALIZED LONG-CHAIN HYDROCARBON MONO- AND DI-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF, AND THEIR USE FOR THE PREVENTION OR TREATMENT OF DISEASE ESPERVITA THERAPEUTICS, INC. 2023-04-13 US claimed
WO-2022159808-A2 FUNCTIONALIZED LONG-CHAIN HYDROCARBON MONO- AND DI-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF, AND THEIR USE FOR THE PREVENTION OR TREATMENT OF DISEASE ESPERVITA THERAPEUTICS, INC. (US) 2022-07-28 WO claimed
WO-2022159811-A1 FUNCTIONALIZED LONG-CHAIN HYDROCARBON MONO- AND DI-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF, AND THEIR USE FOR THE PREVENTION OR TREATMENT OF DISEASE ESPERVITA THERAPEUTICS, INC. (US) 2022-07-28 WO claimed
EP-4003314-A1 FUNCTIONALIZED LONG-CHAIN HYDROCARBON MONO- AND DI-CARBOXYLIC ACIDS USEFUL FOR THE PREVENTION OR TREATMENT OF DISEASE Espervita Therapeutics, Inc. (US) 2022-06-01 EP claimed
WO-2022087173-A1 PHOSPHAPLATIN COMPOUNDS AS THERAPEUTIC AGENTS SELECTIVELY TARGETING HIGHLY GLYCOLYTIC TUMOR CELLS AND METHODS THEREOF PHOSPLATIN THERAPEUTICS INC. (US) 2022-04-28 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230113853-A1 FUNCTIONALIZED LONG-CHAIN HYDROCARBON MONO- AND DI-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF, AND THEIR USE FOR THE PREVENTION OR TREATMENT OF DISEASE AHR, PKD1, CFTR ALDH1A1 180/4885LTC4S 688/4885RAB9A 3842/4885
US-20230144846-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OXER1, OCIAD1, OCIAD2 ALDH1A1 501/4885LTC4S 398/4885RAB9A 819/4885
US-20240009212-A1 PHOSPHAPLATIN COMPOUNDS AS THERAPEUTIC AGENTS SELECTIVELY TARGETING HIGHLY GLYCOLYTIC TUMOR CELLS AND METHODS THEREOF PHGDH, HIF1A, HIF1AN ALDH1A1 865/4885LTC4S 4125/4885RAB9A 2253/4885
US-20230111520-A1 FUNCTIONALIZED LONG-CHAIN HYDROCARBON MONO- AND DI-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF, AND THEIR USE FOR THE PREVENTION OR TREATMENT OF DISEASE CPT1A, PPARG, PC ALDH1A1 288/4885LTC4S 1086/4885RAB9A 4161/4885
US-20240251654-A1 ORGANIC ELECTROLUMINESCENT DEVICE LEF1, EFNA1, EML4 ALDH1A1 131/4885LTC4S 943/4885RAB9A 2013/4885
US-20240317787-A1 ORGANIC ELECTROLUMINESCENT DEVICE EPCAM, ORC3, OCIAD1 ALDH1A1 130/4885LTC4S 2686/4885RAB9A 2646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.