SCHEMBL2945375

SCHEMBL2945375

COc1cc(C=Cc2ccccc2)ccc1O

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.75
TUBB1 Q9H4B7 2/20 0.75
APP P05067 5/20 0.73
MAPT P10636 1/20 0.73
TTR P02766 1/20 0.72
CYP1A2 P05177 2/20 0.71
CYP1A1 P04798 1/20 0.71
CYP1B1 Q16678 1/20 0.71
TYR P14679 1/20 0.69
ALOX5 P09917 2/20 0.68
KDM4E B2RXH2 1/20 0.66
CA12 O43570 1/20 0.66
CA1 P00915 1/20 0.66
CA2 P00918 1/20 0.66
CA3 P07451 1/20 0.66
PKM P14618 1/20 0.66
CSNK2A2 P19784 1/20 0.66
CA4 P22748 1/20 0.66
CA6 P23280 1/20 0.66
CA5A P35218 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2534835 1.00 NFE2L2 (0.75) NFE2L2TUBB1APPMAPTTTR
SCHEMBL4938984 1.00 NFE2L2 (0.75) NFE2L2TUBB1APPMAPTTTR
Isoeugenol SCHEMBL2686818 0.92 TYR (0.84) NFE2L2TUBB1APPMAPTTTR
Cis/Trans-Isoeugenol SCHEMBL2686822 0.92 TYR (0.84) NFE2L2TUBB1APPMAPTTTR
SCHEMBL17732299 0.91 TTR (0.85) NFE2L2APPMAPTTTRCYP1A2
SCHEMBL671150 0.91 TTR (0.85) NFE2L2APPMAPTTTRCYP1A2
SCHEMBL30807100 0.91 TTR (0.85) NFE2L2APPMAPTTTRCYP1A2
SCHEMBL671149 0.91 TTR (0.85) NFE2L2APPMAPTTTRCYP1A2
SCHEMBL5598747 0.88 CYP2D6 (0.85) NFE2L2APPMAPTCYP1A2TYR
Ferulate SCHEMBL28581353 0.88 KDM4E (0.88) NFE2L2APPMAPTCYP1A2TYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080139650-A1 Fungicidally Active Polymer Dispersions And Use Thereof CELANESE EMULSIONS GMBH (DE) 2008-06-12 US claimed
CN-110187119-B Methods and compositions for the detection and treatment of preeclampsia 耶鲁大学 2022-07-29 CN disclosed
CN-110187121-B Methods and compositions for the detection and treatment of preeclampsia 耶鲁大学 2022-07-01 CN disclosed
CN-110187120-B Methods and compositions for the detection and treatment of preeclampsia 耶鲁大学 2022-07-01 CN disclosed
CN-111936628-A Alzheimer disease animal model and application thereof 清华大学 2020-11-13 CN disclosed
US-9925153-B2 Therapeutic agents for skin diseases and conditions STC.UNM (US) 2018-03-27 US disclosed
US-20160287531-A1 THERAPEUTIC AGENTS FOR SKIN DISEASES AND CONDITIONS STC.UNM 2016-10-06 US disclosed
US-8980954-B2 Substituted cis- and trans-stilbenes as therapeutic agents STC.UNM (US) 2015-03-17 US disclosed
US-8716532-B2 One pot multicomponent synthesis of some novel hydroxy stilbene derivatives with alpha, beta-carbonyl conjugation under microwave irradiation COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2014-05-06 US disclosed
US-20130178536-A1 SUBSTITUTED CIS- AND TRANS-STILBENES AS THERAPEUTIC AGENTS STC.UNM (US) 2013-07-11 US disclosed
US-20120165567-A1 ONE POT MULTICOMPONENT SYNTHESIS OF SOME NOVEL HYDROXY STILBENE DERIVATIVES WITH ALPHA, BETA-CARBONYL CONJUGATION UNDER MICROWAVE IRRADIATION COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2012-06-28 US disclosed
WO-2010113005-A2 ONE POT MULTICOMPONENT SYNTHESIS OF SOME NOVEL HYDROXY STILBENE DERIVATIVES WITH ALPHA, BETA-CARBONYL CONJUGATION UNDER MICROWAVE IRRADIATION COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2010-10-07 WO disclosed
US-7759527-B2 Microwave induced one pot process for the preparation of arylethenes COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2010-07-20 US disclosed
US-20080139650-A1 Fungicidally Active Polymer Dispersions And Use Thereof CELANESE EMULSIONS GMBH (DE) 2008-06-12 US disclosed
US-20080045752-A1 Microwave Induced One Pot Process For The Preparation Of Arylethenes COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2008-02-21 US disclosed
US-20070249647-A1 Substituted CIS- and trans-stilbenes as therapeutic agents REGENTS OF THE UNIVERSITY OF NEW MEXICO 2007-10-25 US disclosed
WO-2007110881-A1 A MICROWAVE INDUCED ONE POT PROCESS FOR THE PREPARATION OF ARYLETHENES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2007-10-04 WO disclosed
US-5977105-A Compounds ASTRA PHARMAEUTICALS LTD. (GB) 1999-11-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045752-A1 Microwave Induced One Pot Process For The Preparation Of Arylethenes TET2, HCN4, KDM4E NFE2L2 732/4885TUBB1 1384/4885APP 3839/4885
US-20160287531-A1 THERAPEUTIC AGENTS FOR SKIN DISEASES AND CONDITIONS CUTA, TSLP, ELANE NFE2L2 696/4885TUBB1 15/4885APP 475/4885
US-20120165567-A1 ONE POT MULTICOMPONENT SYNTHESIS OF SOME NOVEL HYDROXY STILBENE DERIVATIVES WITH ALPHA, BETA-CARBONYL CONJUGATION UNDER MICROWAVE IRRADIATION SIK1, SIK2, HCK NFE2L2 237/4885TUBB1 374/4885APP 2941/4885
US-20080139650-A1 Fungicidally Active Polymer Dispersions And Use Thereof CBR3, CBR1, CYP3A4 NFE2L2 3306/4885TUBB1 348/4885APP 3335/4885
US-20070249647-A1 Substituted CIS- and trans-stilbenes as therapeutic agents TGFB1, VHL, TMSB10 NFE2L2 68/4885TUBB1 33/4885APP 546/4885
US-20130178536-A1 SUBSTITUTED CIS- AND TRANS-STILBENES AS THERAPEUTIC AGENTS PSEN1, TERT, PSEN2 NFE2L2 63/4885TUBB1 120/4885APP 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.