SCHEMBL29555

SCHEMBL29555

Fc1ccc(OC2CC2)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 3/20 0.43
GRIN2B Q13224 3/20 0.43
GPR6 P46095 11/20 0.42
CYP2D6 P10635 5/20 0.42
SLC6A2 P23975 2/20 0.41
SLC6A3 Q01959 2/20 0.41
HTR1A P08908 1/20 0.41
TYRO3 Q06418 1/20 0.40
TRPA1 O75762 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26144164 0.90 CSNK2A1 (0.41) GRIN1GRIN2BGPR6CYP2D6
SCHEMBL3115490 0.87 GPR6 (0.41) GRIN1GRIN2BGPR6CYP2D6
SCHEMBL941030 0.87 SLC6A2 (0.58) SLC6A2SLC6A3HTR1ASLC6A4
Hydrochloric Acid SCHEMBL2778482 0.86 SLC6A2 (0.56) SLC6A2SLC6A3HTR1ASLC6A4
SCHEMBL19262515 0.84 GPR6 (0.51) GPR6CYP2D6
SCHEMBL2299176 0.82 GRIN1 (0.40) GRIN1GRIN2BGPR6CYP2D6TRPA1
SCHEMBL14956969 0.82 SLC6A4 (0.59) SLC6A2SLC6A3HTR1ASLC6A4
SCHEMBL31471467 0.81 GRIN1 (0.42) GRIN1GRIN2BGPR6TRPA1SLC6A4
SCHEMBL31471369 0.81 GRIN1 (0.48) GRIN1GRIN2BGPR6CYP2D6TRPA1
Hydrochloric Acid SCHEMBL30357915 0.81 SLC6A4 (0.57) SLC6A2SLC6A3HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704118-B1 AMINOIMIDAZOPYRIDAZINES AS KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-01-12 EP disclosed
US-9241487-B2 Pyrimidine derivatives and use thereof as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-26 US disclosed
US-9198429-B2 Heterocyclic alkanol-derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-12-01 US disclosed
US-9095136-B2 2-IODO imidazole-derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-04 US disclosed
EP-2609088-B1 5-IODO-TRIAZOLE DERIVATIVES BAYER IP GMBH (DE) 2015-04-29 EP disclosed
US-8969248-B2 5-iodotriazole derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-03-03 US disclosed
US-20140336232-A1 2-IODO IMIDAZOLE-DERIVATIVES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-11-13 US disclosed
EP-2782904-A1 NOVEL HETEROCYCLIC ALKANOL-DERIVATIVES Bayer Intellectual Property GmbH (DE) 2014-10-01 EP disclosed
US-20140274952-A1 NOVEL HETEROCYCLIC ALKANOL-DERIVATIVES BAYER INTELLCTUAL PROPERTY GMBH (DE) 2014-09-18 US disclosed
US-20140031373-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS PESTICIDES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-01-30 US disclosed
EP-2646418-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS PESTICIDES Bayer Intellectual Property GmbH (DE) 2013-10-09 EP disclosed
EP-2609088-A1 5-IODO-TRIAZOLE DERIVATIVES Bayer Intellectual Property GmbH (DE) 2013-07-03 EP disclosed
WO-2013076227-A1 NOVEL HETEROCYCLIC ALKANOL-DERIVATIVES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-05-30 WO disclosed
US-20120220638-A1 5-Iodotriazole derivatives BAYER CROPSCIENCE AG (DE) 2012-08-30 US disclosed
WO-2012072547-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-06-07 WO disclosed
WO-2012025506-A1 5-IODO-TRIAZOLE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2012-03-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140336232-A1 2-IODO IMIDAZOLE-DERIVATIVES CIP2A, ING2, AZI2 GRIN1 2910/4885GRIN2B 3113/4885GPR6 4586/4885
US-20140031373-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS PESTICIDES TYMP, TYMS, UMPS GRIN1 2890/4885GRIN2B 3096/4885GPR6 3682/4885
US-20120220638-A1 5-Iodotriazole derivatives INMT, IGFBP5, HDHD5 GRIN1 2132/4885GRIN2B 2403/4885GPR6 4678/4885
US-20140274952-A1 NOVEL HETEROCYCLIC ALKANOL-DERIVATIVES ERG28, CBR3, MYB GRIN1 4072/4885GRIN2B 4333/4885GPR6 4173/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.