SCHEMBL29561

SCHEMBL29561

COc1c2ccc(Cl)cc2c(OC)c2occc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.53
CYP1A1 P04798 4/20 0.53
CYP1A2 P05177 4/20 0.53
CYP1B1 Q16678 4/20 0.53
HPGD P15428 2/20 0.53
KDM4E B2RXH2 2/20 0.53
POLB P06746 1/20 0.53
ABCB11 O95342 1/20 0.49
ALDH1A1 P00352 3/20 0.48
ALOX15 P16050 1/20 0.48
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
PDE4A P27815 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KCNA2 P16389 2/20 0.43
KCNA4 P22459 1/20 0.43
KCNA5 P22460 1/20 0.43
KCNA1 Q09470 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111 0.79 ALDH1A1 (0.60) CYP3A4CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL602977 0.77 KDM4E (0.62) KDM4EPOLBABCB11ALDH1A1MAPK1
SCHEMBL30043104 0.77 KDM4E (0.62) KDM4EPOLBABCB11ALDH1A1MAPK1
SCHEMBL29368971 0.77 KDM4E (0.62) KDM4EPOLBABCB11ALDH1A1MAPK1
Isopimpinellin SCHEMBL498907 0.69 CYP3A4 (1.00) CYP3A4CYP1A1CYP1A2CYP1B1HPGD
Isopimpinellin SCHEMBL29568822 0.69 CYP3A4 (1.00) CYP3A4CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL21297326 0.67 ABCB11 (0.56) KDM4EABCB11ALDH1A1MAPK1SMN1; SMN2
Lonapalene SCHEMBL120134 0.66 ABCB11 (1.00) CYP1A2HPGDKDM4EPOLBABCB11
SCHEMBL6008826 0.65 ABCB11 (0.53) ABCB11CYP2A6
Pimpinellin SCHEMBL2255899 0.65 CYP3A4 (1.00) CYP3A4CYP1A1CYP1A2CYP1B1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103153975-B Novel naphthoquinones for use in the treatment of disease Hangzhou Yier Biological Technology Co.,Ltd. (CN) 2016-01-20 CN disclosed
US-8871802-B2 Naphthoquinones for disease therapies ZHOUSHAN HAIZHONGZHOU XINSHENG PHARMACEUTICALS CO., LTD. (CN) 2014-10-28 US disclosed
US-20130150437-A1 NAPHTHOQUINONES FOR DISEASE THERAPIES ZHOUSHAN HAIZHONGZHOU XINSHENG PHARMACEUTICALS CO., LTD. (CN) 2013-06-13 US disclosed
WO-2012024818-A1 NOVEL ANPHTHOQUINONES FOR DISEASE THERAPIES ZHOUSHAN HAIZHONGZHOU XINSHENG PHARMACEUTICALS CO., LTD. (CN) 2012-03-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130150437-A1 NAPHTHOQUINONES FOR DISEASE THERAPIES NQO1, NME2, CYP27B1 CYP3A4 2063/4885CYP1A1 437/4885CYP1A2 495/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.