SCHEMBL29856346

SCHEMBL29856346

CCc1c(C=O)c2ccnc(OC)c2n1C

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 7/20 0.34
MAOA P21397 1/20 0.34
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
ACSS2 Q9NR19 1/20 0.32
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
HASPIN Q8TF76 3/20 0.30
DYRK2 Q92630 1/20 0.30
MTNR1A P48039 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29856229 0.73 ALOX15 (0.39) CYP3A4HPGD
SCHEMBL29857005 0.69 SLC22A12 (0.43) CYP1A2CYP3A4HPGDCYP2C19
SCHEMBL22863572 0.69 ALDH1A1 (0.46) DYRK1AMAOABCHEACHEDDB1
SCHEMBL29856253 0.68 ERN1 (0.35) ACSS2CYP1A2CYP3A4HPGDCYP2C19
SCHEMBL441518 0.65 ERN1 (0.37) MAOA
SCHEMBL746493 0.65 ERN1 (0.44)
SCHEMBL29954802 0.65 ERN1 (0.37) MAOA
SCHEMBL29856468 0.64 ACSS2 (0.38) DYRK1AMAOABCHEACHEACSS2
SCHEMBL25230147 0.63 ERN1 (0.36) CYP3A4CYP2C19
SCHEMBL772591 0.63 ERN1 (0.46) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022169974-A1 INHIBITORS OF URAT1 AND PHARMACEUTICAL USES THEREOF NEXYS THERAPEUTICS, INC. (US) 2022-08-11 WO disclosed