SCHEMBL299079

SCHEMBL299079

O=C1COc2ccc(Br)cc2N1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.65
PARP1 P09874 3/20 0.59
ALDH1A1 P00352 6/20 0.56
KMT2A Q03164 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
MAPT P10636 4/20 0.54
CMA1 P23946 1/20 0.51
AHR P35869 1/20 0.51
PKM P14618 2/20 0.51
GAA P10253 2/20 0.50
PDE3B Q13370 1/20 0.50
PDE3A Q14432 1/20 0.50
NR3C2 P08235 3/20 0.49
HPGD P15428 1/20 0.49
BRAF P15056 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29452973 1.00 MMP12 (0.65) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL305202 0.86 MMP12 (0.51) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL30336661 0.86 MMP12 (0.51) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL15964650 0.83 CMA1 (0.49) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL30896836 0.83 CMA1 (0.49) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL8195292 0.80 MMP12 (0.41) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL302933 0.79 MMP12 (0.65) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL707058 0.79 MMP12 (0.65) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL279594 0.79 MMP12 (1.00) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL8184077 0.79 MMP12 (0.65) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 399 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078131-A1 PYRROLO-PYRIDAZINE INHIBITORS OF JAK2 AJAX THERAPEUTICS INC (US) 2026-03-19 US disclosed
US-12545653-B2 Compound as PPAR agonist and application thereof USA Elixiria Biotech Inc. (US) 2026-02-10 US disclosed
WO-2025235763-A1 FLUORESCENT PROBES AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-11-13 WO disclosed
US-12275723-B2 Compounds and uses thereof JANSSEN PHARMACEUTICA NV (BE) 2025-04-15 US disclosed
US-20240400546-A1 COMPOUNDS AND USES THEREOF JANSSEN PHARMACEUTICA NV (BE) 2024-12-05 US disclosed
US-20240400499-A1 NOVEL AMINO ACID DERIVATIVES PEPTIDREAM INC (JP) 2024-12-05 US disclosed
US-20240300938-A1 COMPOUNDS AND USES THEREOF JANSSEN PHARMACEUTICA NV (BE) 2024-09-12 US disclosed
CN-114436955-B Tetrahydroquinoline and benzomorpholine derivatives or salts thereof, and preparation method and application thereof 复旦大学 2024-08-09 CN disclosed
CN-115677611-B 2H-benzo [ b ] [1,4] oxazin-3 (4H) -one derivatives 成都硕德药业有限公司 2024-07-09 CN disclosed
US-11970486-B2 Compounds and uses thereof JANSSEN PHARMACEUTICA NV (BE) 2024-04-30 US disclosed
US-20050014938-A1 Phenyl substituted triazoles and their use as selective inhibitors of akl5 kinase GASTER LARAMIE MARY (GB) 2005-01-20 US disclosed
US-20040266842-A1 Thiazolyl substituted triazoles as alk5 inhibitors GASTER LARAMIE MARY 2004-12-30 US disclosed
EP-1444227-A1 THIAZOLYL SUBSTITUTED TRIAZOLES AS ALK5 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-08-11 EP disclosed
WO-2004046124-A1 BENZOXAZINONE DERIVATIVES, PREPARATION THEREOF AND USES IN THE TREATMENT OF CNS AND OTHER DISORDERS GLAXO GROUP LIMITED (GB) 2004-06-03 WO disclosed
US-20040092512-A1 Substituted benzoxazinones and uses thereof ROCHE PALO ALTO LLC 2004-05-13 US disclosed
US-20040063704-A1 Benzoxazinone derivatives, their preparation and use SMITHKLINE BEECHAM P.L.C (GB) 2004-04-01 US disclosed
EP-1330460-A2 BENZOXAZINONE DERIVATIVES, THEIR PREPARATION AND USE SMITHKLINE BEECHAM PLC (GB) 2003-07-30 EP disclosed
WO-2003042207-A1 THIAZOLYL SUBSTITUTED TRIAZOLES AS ALK5 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-05-22 WO disclosed
WO-2002034754-A2 BENZOXAZINONE DERIVATIVES, THEIR PREPARATION AND USE SMITHKLINE BEECHAM P.L.C. (GB) 2002-05-02 WO disclosed
US-5141935-A Dihydrobenz thiazine derivative and microorganism control agent UBE INDUSTRIES, LTD. (JP) 1992-08-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12545653-B2 Compound as PPAR agonist and application thereof PPARA, PPARD, PPARG MMP12 2439/4885PARP1 2679/4885ALDH1A1 784/4885
US-20040063704-A1 Benzoxazinone derivatives, their preparation and use CYP2B6, CBR1, CYP2A6 MMP12 3044/4885PARP1 865/4885ALDH1A1 1181/4885
US-20260078131-A1 PYRROLO-PYRIDAZINE INHIBITORS OF JAK2 JAK2, JAK1, JAK3 MMP12 3089/4885PARP1 1838/4885ALDH1A1 2846/4885
US-20240300938-A1 COMPOUNDS AND USES THEREOF NLN, ACHE, CLN6 MMP12 1820/4885PARP1 1952/4885ALDH1A1 656/4885
US-20050014938-A1 Phenyl substituted triazoles and their use as selective inhibitors of akl5 kinase AKR1C3, CBR3, PHKG1 MMP12 4730/4885PARP1 2165/4885ALDH1A1 2451/4885
US-20040266842-A1 Thiazolyl substituted triazoles as alk5 inhibitors CBR3, CBR1, ALK MMP12 4826/4885PARP1 1393/4885ALDH1A1 1905/4885
US-20240400546-A1 COMPOUNDS AND USES THEREOF NLN, ACHE, CLN6 MMP12 1820/4885PARP1 1952/4885ALDH1A1 656/4885
US-12275723-B2 Compounds and uses thereof NLN, ACHE, CLN6 MMP12 1820/4885PARP1 1952/4885ALDH1A1 656/4885
US-20040092512-A1 Substituted benzoxazinones and uses thereof CYP4X1, CYP3A5, CYP2D6 MMP12 2222/4885PARP1 488/4885ALDH1A1 389/4885
US-20240400499-A1 NOVEL AMINO ACID DERIVATIVES BCAT1, BCAT2, PELP1 MMP12 4236/4885PARP1 4794/4885ALDH1A1 4472/4885
US-11970486-B2 Compounds and uses thereof NLN, ACHE, CLN6 MMP12 1820/4885PARP1 1952/4885ALDH1A1 656/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.