SCHEMBL305202

SCHEMBL305202

O=C1COc2cc(Br)ccc2N1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.51
CYP11B1 P15538 2/20 0.51
CYP11B2 P19099 2/20 0.51
PDE3B Q13370 1/20 0.50
PDE3A Q14432 1/20 0.50
PARP1 P09874 1/20 0.47
CMA1 P23946 1/20 0.47
AHR P35869 1/20 0.47
KIF11 P52732 1/20 0.47
DRD4 P21917 6/20 0.46
DRD3 P35462 6/20 0.46
DRD2 P14416 5/20 0.46
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HTR1A P08908 1/20 0.44
CHRM5 P08912 1/20 0.44
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30336661 1.00 MMP12 (0.51) MMP12CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL299079 0.86 MMP12 (0.65) MMP12PDE3BPDE3APARP1CMA1
SCHEMBL29452973 0.86 MMP12 (0.65) MMP12PDE3BPDE3APARP1CMA1
SCHEMBL24720317 0.83 CMA1 (0.45) CYP11B1CYP11B2PDE3BPDE3ACMA1
SCHEMBL30053776 0.79 NR3C2 (0.57) MMP12CYP11B1CYP11B2PARP1KIF11
SCHEMBL3594625 0.79 MMP12 (0.51) MMP12CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL1861248 0.79 NR3C2 (0.57) MMP12CYP11B1CYP11B2PARP1KIF11
SCHEMBL30799148 0.79 MMP12 (0.51) MMP12CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL276741 0.79 MMP12 (0.51) MMP12CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL304249 0.79 DRD4 (0.56) MMP12CYP11B1CYP11B2PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 139 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078117-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS INC (US) 2026-03-19 US disclosed
EP-4696688-A1 BENZO-FUSED RING COMPOUND INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2026-02-18 EP disclosed
US-20260015321-A1 CHEMICAL COMPOUNDS AND USES THEREOF GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.4) LIMITED (GB) 2026-01-15 US disclosed
EP-4663630-A1 NOVEL BENZIMIDAZOLONE DERIVATIVE COMPOUND AS AUTOTAXIN INHIBITOR LG Chem, Ltd. (KR) 2025-12-17 EP disclosed
US-20250340529-A1 Heterocyclic Compounds as Immunomodulators of PD-L1 Interactions ASCLETIS BIOSCIENCE CO LTD (CN) 2025-11-06 US disclosed
WO-2025201477-A1 SPIROCYCLIC GSDME INHIBITORS PYROTECH (BEIJING) BIOTECHNOLOGY CO.,LTD. (CN) 2025-10-02 WO disclosed
EP-4624464-A1 PYRIDINE POLYCYCLIC COMPOUND INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2025-10-01 EP disclosed
US-20250205219-A1 TARGETED DEGRADATION OF VAV1 MONTE ROSA THERAPEUTICS AG (CH) 2025-06-26 US disclosed
US-12304907-B2 Compounds and methods of use TANGO THERAPEUTICS, INC. (US) 2025-05-20 US disclosed
US-12275723-B2 Compounds and uses thereof JANSSEN PHARMACEUTICA NV (BE) 2025-04-15 US disclosed
US-20080221093-A1 Metalloprotease inhibitors containing a heterocyclic moiety ALANTOS PHARMACEUTICALS HOLDING, INC. 2008-09-11 US disclosed
US-20080221093-A1 Metalloprotease inhibitors containing a heterocyclic moiety ALANTOS PHARMACEUTICALS HOLDING, INC. 2008-09-11 US disclosed
WO-2008001076-A1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2008-01-03 WO disclosed
EP-1196412-B1 NITROGEN CONTAINING HETEROBICYCLES AS FACTOR XA INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2004-06-09 EP disclosed
US-6716841-B2 SUCH AS 1-((1-(3-(AMINOMETHYL)PHENYL)-3-(TRIFLUOROMETHYL)-1H-PYRAZOL-5-YL)CARBONYL) -5-(2-( AMINOSULFONYL)PHENYL)-2,3-DIHYDRO-1H-INDOLE FOR TREATMENT AND PREVENTION OF THROMBOEMBOLIC DISORDERS; ANTICOAGULANTS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-04-06 US disclosed
US-20030096820-A1 Nitrogen containing heterobicycles as factor Xa inhibitors JACOBSON IRINA C (US) 2003-05-22 US disclosed
US-6534535-B1 Administering indole derivative as anticoagulant MILLENNIUM PHARMACEUTICALS, INC. 2003-03-18 US disclosed
WO-2001012600-A9 INHIBITORS OF FACTOR Xa COR THERAPEUTICS INC (US) 2002-09-12 WO disclosed
US-6429205-B1 ANTICOAGULANTS BRISTOL-MEYERS SQUIBB PHARMA COMPANY 2002-08-06 US disclosed
WO-2001012600-A1 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2001-02-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030096820-A1 Nitrogen containing heterobicycles as factor Xa inhibitors SERPINC1, CTRB1, F2 MMP12 679/4885CYP11B1 1202/4885CYP11B2 2168/4885
US-20250340529-A1 Heterocyclic Compounds as Immunomodulators of PD-L1 Interactions CD274, PDCD1LG2, PDCD1 MMP12 707/4885CYP11B1 1746/4885CYP11B2 1568/4885
US-12275723-B2 Compounds and uses thereof NLN, ACHE, CLN6 MMP12 1820/4885CYP11B1 192/4885CYP11B2 93/4885
US-20260015321-A1 CHEMICAL COMPOUNDS AND USES THEREOF WRN, MSH2, MSH6 MMP12 2677/4885CYP11B1 2743/4885CYP11B2 2880/4885
US-20080221093-A1 Metalloprotease inhibitors containing a heterocyclic moiety MMP12, MMP13, MMP25 MMP12 1/4885CYP11B1 565/4885CYP11B2 675/4885
US-12304907-B2 Compounds and methods of use F12, C1R, ABCG2 MMP12 4148/4885CYP11B1 68/4885CYP11B2 86/4885
US-20250205219-A1 TARGETED DEGRADATION OF VAV1 VAV1, KRAS, CBL MMP12 1036/4885CYP11B1 4229/4885CYP11B2 4345/4885
US-20260078117-A1 COMPOUNDS AND METHODS OF USE NR3C2, ADRA1A, CNR1 MMP12 3729/4885CYP11B1 104/4885CYP11B2 92/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.