SCHEMBL2999130

SCHEMBL2999130

O=C(CBr)c1ccccc1OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SGMS2 Q8NHU3 5/20 0.59
NPC1 O15118 1/20 0.56
HTT P42858 1/20 0.56
GAA P10253 1/20 0.55
FOLH1 Q04609 1/20 0.54
PARP1 P09874 1/20 0.53
L3MBTL1 Q9Y468 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
ALDH1A1 P00352 1/20 0.52
PTGER1 P34995 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30194507 1.00 SGMS2 (0.59) SGMS2NPC1HTTGAAFOLH1
SCHEMBL20819560 0.86 NPC1 (0.53) SGMS2NPC1HTTGAAFOLH1
SCHEMBL4481452 0.85 FFAR4 (0.51) SGMS2NPC1FOLH1L3MBTL1LMNA
SCHEMBL3679181 0.85 SGMS2 (0.60) SGMS2NPC1HTTGAAFOLH1
SCHEMBL4473413 0.84 MAOB (0.61) NPC1FOLH1MEN1KMT2ALMNA
SCHEMBL14339650 0.83 SGMS2 (0.59) SGMS2NPC1HTTGAAFOLH1
SCHEMBL4431127 0.83 SGMS2 (0.59) SGMS2NPC1HTTGAAPARP1
SCHEMBL6243854 0.83 NPC1 (0.64) SGMS2NPC1HTTGAAPARP1
SCHEMBL19156329 0.83 SGMS2 (0.59) SGMS2NPC1HTTGAAFOLH1
SCHEMBL4944383 0.83 NPC1 (0.60) SGMS2NPC1HTTGAAFOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 101 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3672582-B1 COMPOSITIONS AND METHODS FOR TREATING CANCER CEDARS SINAI MEDICAL CENTER (US) 2026-04-15 EP disclosed
US-20260015316-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER CEDARS-SINAI MEDICAL CENTER (US) 2026-01-15 US disclosed
US-12421185-B2 Compositions and methods for treating cancer CEDARS-SINAI MEDICAL CENTER (US) 2025-09-23 US disclosed
US-20250145598-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF UNIV CALIFORNIA (US) 2025-05-08 US disclosed
US-20250064945-A1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE GENENTECH, INC. 2025-02-27 US disclosed
EP-4436965-A1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE Arvinas Operations, Inc. (US) 2024-10-02 EP disclosed
EP-4387617-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF The Regents of the University of California (US) 2024-06-26 EP disclosed
WO-2023096987-A1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. (US) 2023-06-01 WO disclosed
WO-2023096987-A1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. (US) 2023-06-01 WO disclosed
WO-2023023156-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-02-23 WO disclosed
US-5877193-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 1999-03-02 US disclosed
EP-0882707-A1 NOVEL TRICYCLIC COMPOUNDS AND DRUG COMPOSITIONS CONTAINING THE SAME Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1998-12-09 EP disclosed
EP-0819681-A2 N-(4-Aryl-thiazol-2-yl)-sulfonamides and their use F. HOFFMANN-LA ROCHE AG (CH) 1998-01-21 EP disclosed
EP-0647632-A1 NOVEL BENZODIAZEPINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-04-12 EP disclosed
EP-0428423-A2 Aryloxy alkyl benzenes, processes for their preparation and pharmaceutical compositions containing them LIPHA S.A. (FR) 1991-05-22 EP disclosed
EP-0037062-B1 SUBSTITUTED 3-ARYL-2-CYCLOALKENE-1-ONES, PROCESS FOR THEIR PREPARATION AND THEIR PARMACEUTICAL USE Beiersdorf Aktiengesellschaft (DE) 1984-10-17 EP disclosed
US-4401831-A ADRENOLYTIC AND HYPOTENSIVE AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1983-08-30 US disclosed
US-4358460-A HYPOTENSIVE, ANTIARRHYTHMIA, ANGINA PECTORIS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1982-11-09 US disclosed
EP-0037062-A2 Substituted 3-aryl-2-cycloalkene-1-ones, process for their preparation and their parmaceutical use Beiersdorf Aktiengesellschaft (DE) 1981-10-07 EP disclosed
US-4265903-A HYPOTENSIVE, ADRENOLYTIC BEIERSDORF AKTIENGESELLSCHAFT (DE) 1981-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250145598-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF ASAH2, ASAH1, ACER2 SGMS2 225/4885NPC1 340/4885HTT 4119/4885
US-12421185-B2 Compositions and methods for treating cancer TSG101, RNASE1, TP53 SGMS2 416/4885NPC1 638/4885HTT 2878/4885
US-20250064945-A1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE ADRM1, BRAP, VHL SGMS2 3508/4885NPC1 2270/4885HTT 640/4885
US-20260015316-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER GLI1, RCC2, BRCA1 SGMS2 1600/4885NPC1 356/4885HTT 1185/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.