SCHEMBL30003076

SCHEMBL30003076

CC(C(=O)c1ccccc1)c1nc(-c2ccccc2)co1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
HTR2A P28223 1/20 0.40
HRH1 P35367 1/20 0.40
KCNH2 Q12809 1/20 0.40
DAGLA Q9Y4D2 1/20 0.39
ADORA1 P30542 6/20 0.39
ADORA3 P0DMS8 3/20 0.39
ADORA2A P29274 3/20 0.39
ENPP3 O14638 2/20 0.38
ENPP1 P22413 2/20 0.38
HSD11B1 P28845 1/20 0.38
ADORA2B P29275 1/20 0.37
SMO Q99835 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6668389 0.78 ENPP3 (0.43) DAGLAADORA1ENPP3ENPP1HSD11B1
SCHEMBL10052155 0.77 ENPP3 (0.45) DAGLAADORA1ADORA3ADORA2AENPP3
SCHEMBL21180807 0.74 ENPP3 (0.43) DAGLAENPP3ENPP1HSD11B1TDP1
SCHEMBL30765909 0.74 ENPP3 (0.43) DAGLAADORA1ADORA2AENPP3ENPP1
SCHEMBL9441037 0.73 MAOA (0.45) ADORA3SMOLMNASMN1; SMN2
SCHEMBL13848629 0.72 ENPP3 (0.44) DAGLAADORA1ADORA3ADORA2AENPP3
SCHEMBL4737344 0.72 MAPT (0.49) TDP1ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL13744630 0.70 ENPP3 (0.42) DAGLAADORA1ADORA3ADORA2AENPP3
SCHEMBL5296166 0.67 DAGLA (0.57) DAGLAENPP3ENPP1HSD11B1SMO
SCHEMBL4806377 0.67 PTGS2 (0.69) PGRADRA2AADRA2BHTR2AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3653613-B1 1,3-DI-SUBSTITUTED KETENE COMPOUND AND APPLICATION THEREOF BEBETTER MED INC (CN) 2022-11-16 EP disclosed