SCHEMBL30296014

SCHEMBL30296014

Cc1onc(-c2cccc(-c3ccccc3COC(C)C)c2S(N)(=O)=O)c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA4 P22748 2/20 0.34
CA7 P43166 2/20 0.34
LMNA P02545 2/20 0.34
CA12 O43570 1/20 0.34
MT-CO2 P00403 1/20 0.34
CA3 P07451 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CHRM1 P11229 1/20 0.34
ADRA2B P18089 1/20 0.34
PTGS1 P23219 1/20 0.34
CA6 P23280 1/20 0.34
SLC6A2 P23975 1/20 0.34
PDE4A P27815 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30296173 0.88 CA4 (0.36) CA1CA2CA4CA7LMNA
SCHEMBL30295930 0.85 CA1 (0.34) CA1CA2CA4CA7LMNA
SCHEMBL30295791 0.77 PTGS2 (0.50) EDNRBEDNRACA1CA2CA4
SCHEMBL7850632 0.77 PTGS2 (0.50) EDNRBEDNRACA1CA2CA4
SCHEMBL29281012 0.76 EDNRA (0.40) EDNRBEDNRALMNAALDH1A1
SCHEMBL30296099 0.74 NR3C1 (0.38) LMNAFFAR1SCN5ASCN9AALDH1A1
SCHEMBL29280986 0.73 P2RX3 (0.38) EDNRBEDNRA
SCHEMBL30296201 0.72 EDNRA (0.51) EDNRBEDNRA
SCHEMBL30295779 0.71 EDNRB (0.38) EDNRBEDNRACA1CA2CA4
SCHEMBL27968617 0.70 CA2 (0.46) EDNRBEDNRACA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023025277-A1 AROMATIC RING-CONTAINING BIOLOGICAL ANTAGONIST, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2023-03-02 WO disclosed