SCHEMBL3033667

SCHEMBL3033667

Cc1cc(NCCn2cccc2)ccc1-n1cnc2c(N)nc(N)nc21

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 2/20 0.38
PI4K2B Q8TCG2 2/20 0.38
PI4K2A Q9BTU6 2/20 0.38
PI4KB Q9UBF8 2/20 0.38
CDK1 P06493 4/20 0.37
CCNB1 P14635 2/20 0.37
CCNE1 P24864 2/20 0.37
CDK2 P24941 2/20 0.37
CRHR1 P34998 2/20 0.33
TMIGD3 P0DMS9 4/20 0.32
ADORA2A P29274 4/20 0.32
ADORA1 P30542 4/20 0.32
ADORA2B P29275 2/20 0.32
CSNK1D P48730 1/20 0.32
CSNK1E P49674 1/20 0.32
DHFR P00374 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3033663 0.73 DHFR (0.34) DHFR
SCHEMBL4972839 0.70 ALDH1A1 (0.41)
SCHEMBL2951209 0.70 KDM4E (0.42) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL2950165 0.69 TLR7 (0.41) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL3040612 0.68 PI4KA (0.42) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL2951937 0.67 DHFR (0.45) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL2955288 0.67 TLR7 (0.42) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL2952316 0.66 NPC1 (0.51) ADORA2AADORA1ADORA2B
SCHEMBL2953257 0.66 CDK1 (0.42) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL2946546 0.65 PI4KA (0.37) PI4KAPI4K2BPI4K2API4KBCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed