Water

Water

SCHEMBL3036870

O.O=CC(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL8330424 1.00
SCHEMBL809285 0.97
SCHEMBL10487190 0.93
Water SCHEMBL31538171 0.90 THRB (0.32)
SCHEMBL11129024 0.90
Water SCHEMBL11048626 0.88 LMNA (0.36)
SCHEMBL9724351 0.87 LMNA (0.33)
Water SCHEMBL11396324 0.86
SCHEMBL25404599 0.84 LMNA (0.38)
SCHEMBL8189397 0.84 LMNA (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119874465-A New method for synthesizing fluoroalkyl substituted 4,4' -diaminodiphenyl methane compound 海南大学 2025-04-25 CN claimed
CN-119874465-A New method for synthesizing fluoroalkyl substituted 4,4' -diaminodiphenyl methane compound 海南大学 2025-04-25 CN disclosed
EP-3757085-B1 PERFLUORINATED POLYOLS AND THEIR USE FOR THE ENANTIOMERIC SEPARATION OF CHIRAL ANIONS CENTRE NAT RECH SCIENT (FR) 2021-11-10 EP disclosed
EP-3757085-A1 PERFLUORINATED POLYOLS AND THEIR USE FOR THE ENANTIOMERIC SEPARATION OF CHIRAL ANIONS Centre National de la Recherche Scientifique (FR) 2020-12-30 EP disclosed
WO-2020260437-A1 PERFLUORINATED POLYOLS AND THEIR USE FOR THE ENANTIOMERIC SEPARATION OF CHIRAL ANIONS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2020-12-30 WO disclosed
US-20100217007-A1 CHEMICAL PROCESS SYNGENTA CROP PROTECTION, INC. (US) 2010-08-26 US disclosed
EP-1469001-B1 Corroles, including chiral derivatives and the use thereof TECHNION RES & DEV FOUNDATION (IL) 2010-05-05 EP disclosed
EP-1928869-B1 CHEMICAL PROCESS SYNGENTA PARTICIPATIONS AG (CH) 2010-03-17 EP disclosed
EP-1928869-A1 CHEMICAL PROCESS Syngeta Participations AG (CH) 2008-06-11 EP disclosed
WO-2007020460-A1 CHEMICAL PROCESS SYNGENTA PARTICIPATIONS AG (CH) 2007-02-22 WO disclosed
EP-0757690-A4 ELECTRON-DEFICIENT PORPHYRINS AND PROCESSES AND INTERMEDIATES FOR PREPARING SAME UNIV PENNSYLVANIA (US) 1999-06-16 EP disclosed
US-5856515-A Electron-deficient porphyrins and processes and intermediates for preparing same TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1999-01-05 US disclosed
US-5817830-A Pyrrolic compounds TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-10-06 US disclosed
EP-0821686-A4 NOVEL PORPHYRINS AND PORPHYRIN SYNTHESIS TECHNIQUES UNIV PENNSYLVANIA (US) 1998-04-15 EP disclosed
EP-0821686-A1 NOVEL PORPHYRINS AND PORPHYRIN SYNTHESIS TECHNIQUES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-02-04 EP disclosed
EP-0757690-A1 ELECTRON-DEFICIENT PORPHYRINS AND PROCESSES AND INTERMEDIATES FOR PREPARING SAME TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1997-02-12 EP disclosed
US-5599924-A Electron-deficient porphyrins and processes and intermediates for preparing same TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1997-02-04 US disclosed
WO-1996017844-A1 NOVEL PORPHYRINS AND PORPHYRIN SYNTHESIS TECHNIQUES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1996-06-13 WO disclosed
WO-1995029916-A1 ELECTRON-DEFICIENT PORPHYRINS AND PROCESSES AND INTERMEDIATES FOR PREPARING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1995-11-09 WO disclosed
EP-0453398-A2 Nitroenamine derivatives as pesticides CIBA-GEIGY AG (CH) 1991-10-23 EP disclosed