SCHEMBL3065860

SCHEMBL3065860

Cn1cc(B(O)O)ccc1=O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.39
LPL P06858 2/20 0.39
LIPG Q9Y5X9 2/20 0.39
ENPP2 Q13822 4/20 0.38
CA1 P00915 2/20 0.35
KDM4E B2RXH2 1/20 0.35
BRD4 O60885 2/20 0.35
TSHR P16473 1/20 0.34
DYRK1A Q13627 1/20 0.33
IDH1 O75874 1/20 0.33
CREBBP Q92793 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14848266 0.75 BRD4 (0.40) BRD4DYRK1AIDH1
SCHEMBL17643854 0.74 LPL (0.41) CA2LPLLIPGENPP2CA1
SCHEMBL3061389 0.73 BRD4 (0.32) BRD4
SCHEMBL29267567 0.71 BRD4 (0.40) KDM4EBRD4DYRK1AIDH1CREBBP
SCHEMBL7247913 0.70
SCHEMBL27226149 0.69 PTGS2 (0.49) CA2LPLLIPGENPP2CA1
SCHEMBL9281070 0.68 BRD4 (0.36) CA2LPLLIPGENPP2CA1
SCHEMBL12063 0.67
SCHEMBL17522917 0.67
SCHEMBL31334167 0.66 ORAI1 (0.41) ENPP2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 139 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119039234-B Pyridazine amide compound and preparation method and application thereof 中国药科大学 2026-05-15 CN disclosed
EP-4731626-A1 PI3K INHIBITORS AND USE THEREOF Regor Pharmaceuticals, Inc. (US) 2026-04-29 EP disclosed
US-12516059-B2 Pyrazolopyridine compounds and uses thereof INCYTE CORPORATION (US) 2026-01-06 US disclosed
EP-4594318-A1 AKT1 MODULATORS Alterome Therapeutics, Inc. (US) 2025-08-06 EP disclosed
US-12264147-B2 Substituted carboxamides as inhibitors of WDR5 protein-protein binding Propellon Therapeutics Inc. (CA) 2025-04-01 US disclosed
US-20250092040-A1 AKT1 MODULATORS ALTEROME THERAPEUTICS, INC. 2025-03-20 US disclosed
WO-2024260464-A1 PI3K INHIBITORS AND USE THEREOF REGOR PHARMACEUTICALS, INC. (US) 2024-12-26 WO disclosed
CN-119039234-A Pyridazine amide compound and preparation method and application thereof 中国药科大学 2024-11-29 CN disclosed
US-20240383889-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF INCYTE CORPORATION 2024-11-21 US disclosed
CN-113906022-B Pyrazolopyridines and triazolopyridines as A2A/A2B inhibitors 因赛特公司 2024-08-09 CN disclosed
US-20130029984-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, LLC (US) 2013-01-31 US disclosed
US-8344001-B2 Heterocyclic H3 antagonists HIGH POINT PHARMACEUTICALS, LLC (US) 2013-01-01 US disclosed
EP-2166846-B1 INHIBITORS OF JANUS KINASES MERCK SHARP & DOHME (US) 2012-10-17 EP disclosed
US-20100267721-A1 Heterocyclic H3 Antagonists HIGH POINT PHARMACEUTICALS LLC (US) 2010-10-21 US disclosed
US-20100256097-A1 INHIBITORS OF JANUS KINASES MERCK SHARP & DOHME LLC 2010-10-07 US disclosed
US-20100256097-A1 INHIBITORS OF JANUS KINASES MERCK SHARP & DOHME LLC 2010-10-07 US disclosed
US-20100256097-A1 INHIBITORS OF JANUS KINASES MERCK SHARP & DOHME LLC 2010-10-07 US disclosed
EP-2014656-A2 New heteocyclic h3 antagonists TRANSTECH PHARMA (US) 2009-01-14 EP disclosed
WO-2008156726-A1 INHIBITORS OF JANUS KINASES MERCK & CO., INC. (US) 2008-12-24 WO disclosed
WO-2008141119-A2 MODULATORS OF CFTR VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-11-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240383889-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF PDXK, PCK1, PGK1 CA2 3502/4885LPL 1774/4885LIPG 2028/4885
US-12264147-B2 Substituted carboxamides as inhibitors of WDR5 protein-protein binding WDR5, WDR82, WDR1 CA2 3299/4885LPL 4483/4885LIPG 4184/4885
US-20100267721-A1 Heterocyclic H3 Antagonists HRH3, HRH4, HRH2 CA2 763/4885LPL 4714/4885LIPG 4855/4885
US-20100256097-A1 INHIBITORS OF JANUS KINASES JAK2, JAK3, JAK1 CA2 3829/4885LPL 3758/4885LIPG 4127/4885
US-20250092040-A1 AKT1 MODULATORS AKT1S1, AKT1, AKT2 CA2 4577/4885LPL 1555/4885LIPG 766/4885
US-20130029984-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PIK3CA, PIK3CD, PIK3CB CA2 2157/4885LPL 1138/4885LIPG 601/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.