SCHEMBL307422

SCHEMBL307422

O=Cc1cc2nccc(Cl)c2s1

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.40
TDP1 Q9NUW8 1/20 0.32
MCHR1 Q99705 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30496258 1.00 CYP2A6 (0.40) CYP2A6TDP1MCHR1
SCHEMBL10272368 0.79 GRIN2D (0.41) CYP2A6
SCHEMBL3571782 0.79 L3MBTL1 (0.33)
SCHEMBL3571779 0.79 L3MBTL1 (0.33)
SCHEMBL23356001 0.77 GRIN3B (0.44) CYP2A6
SCHEMBL15241358 0.77 CYP2A6 (0.38) CYP2A6
SCHEMBL28375772 0.76 PSMB8 (0.33) CYP2A6TDP1
SCHEMBL26915693 0.76 USP7 (0.30)
SCHEMBL31377751 0.74 CYP2A6 (0.49) CYP2A6
SCHEMBL1847722 0.74 NPC1 (0.43) CYP2A6TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260069602-A1 COMPOUNDS, COMPOSITIONS, AND METHODS ACONCAGUA BIO INC (US) 2026-03-12 US disclosed
US-12404279-B2 Deubiquitinase inhibitors and methods of use thereof MOLECURE S.A. (PL) 2025-09-02 US disclosed
EP-4452984-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF Molecure S.A. (PL) 2024-10-30 EP disclosed
US-20240158412-A1 UBIQUITIN-SPECIFIC PROTEASE 7 (USP7) INHIBITORS AND USES THEREOF FAXIAN THERAPEUTICS, LLC 2024-05-16 US disclosed
EP-4288442-A1 UBIQUITIN-SPECIFIC PROTEASE 7 (USP7) INHIBITORS AND USES THEREOF Faxian Therapeutics, LLC (US) 2023-12-13 EP disclosed
US-20230219973-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF MOLECURE S.A. (PL) 2023-07-13 US disclosed
WO-2023119233-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF MOLECURE S.A. (PL) 2023-06-29 WO disclosed
WO-2023119233-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF MOLECURE S.A. (PL) 2023-06-29 WO disclosed
US-20230172914-A1 BIOMARKER-BASED THERAPEUTIC COMPOSITION WELLMARKER BIO CO., LTD. (KR) 2023-06-08 US disclosed
US-20230172914-A1 BIOMARKER-BASED THERAPEUTIC COMPOSITION WELLMARKER BIO CO., LTD. (KR) 2023-06-08 US disclosed
EP-1781664-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING Methylgene, Inc. (CA) 2007-05-09 EP disclosed
WO-2007026221-A2 IMPROVED METHODS FOR PREPARING BENZOFUSED HETEROARYL AMIDE DERIVATIVES OF THIENOPYRIDINES PFIZER INC. (US) 2007-03-08 WO disclosed
WO-2007026221-A2 IMPROVED METHODS FOR PREPARING BENZOFUSED HETEROARYL AMIDE DERIVATIVES OF THIENOPYRIDINES PFIZER INC. (US) 2007-03-08 WO disclosed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US disclosed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US disclosed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US disclosed
US-20060287343-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE, INC. 2006-12-21 US disclosed
US-20060074056-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. (CA) 2006-04-06 US disclosed
WO-2006010264-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE, INC. (CA) 2006-02-02 WO disclosed
US-20020004511-A1 Thiophene derivatives useful as anticancer agents LUZZIO MICHAEL JOSEPH (US) 2002-01-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020004511-A1 Thiophene derivatives useful as anticancer agents CCNA1, CCNE1, TP53 CYP2A6 1392/4885TDP1 48/4885MCHR1 1707/4885
US-20240158412-A1 UBIQUITIN-SPECIFIC PROTEASE 7 (USP7) INHIBITORS AND USES THEREOF USP7, USP28, USP1 CYP2A6 2779/4885TDP1 914/4885MCHR1 4166/4885
US-20060074056-A1 Inhibitors of VEGF receptor and HGF receptor signaling HGF, MET, FLT1 CYP2A6 4426/4885TDP1 4530/4885MCHR1 377/4885
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling HGF, MET, FLT1 CYP2A6 4426/4885TDP1 4530/4885MCHR1 377/4885
US-20060287343-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING HGF, MET, FLT1 CYP2A6 4426/4885TDP1 4530/4885MCHR1 377/4885
US-20230172914-A1 BIOMARKER-BASED THERAPEUTIC COMPOSITION KRAS, RET, NRAS CYP2A6 4625/4885TDP1 2957/4885MCHR1 4465/4885
US-20230219973-A1 DEUBIQUITINASE INHIBITORS AND METHODS OF USE THEREOF USP7, USP28, USP1 CYP2A6 2548/4885TDP1 876/4885MCHR1 3840/4885
US-12404279-B2 Deubiquitinase inhibitors and methods of use thereof USP7, USP28, USP1 CYP2A6 2548/4885TDP1 876/4885MCHR1 3840/4885
US-20260069602-A1 COMPOUNDS, COMPOSITIONS, AND METHODS SCTR, SSTR1, NPY1R CYP2A6 1020/4885TDP1 1946/4885MCHR1 131/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.