SCHEMBL30747808

SCHEMBL30747808

CCOC(=O)c1ccnc2ccc(F)cc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
NMT2 O60551 1/20 0.55
NMT1 P30419 1/20 0.55
NUDT1 P36639 1/20 0.52
MAPT P10636 4/20 0.52
KDM4E B2RXH2 4/20 0.52
L3MBTL1 Q9Y468 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
GAA P10253 2/20 0.52
ATM Q13315 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.50
LMNA P02545 2/20 0.50
ALDH1A1 P00352 4/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
MAPK1 P28482 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
POLB P06746 1/20 0.44
NPC1 O15118 1/20 0.44
ALPL P05186 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30747811 0.89 TSHR (0.54) TSHRNMT2NMT1NUDT1MAPT
SCHEMBL11655288 0.86 KDM4E (0.59) NMT1NUDT1MAPTKDM4EL3MBTL1
SCHEMBL22492342 0.84 PLA2G2A (0.54) KDM4EL3MBTL1LMNA
SCHEMBL31510551 0.83 ALDH1A1 (0.66) TSHRNUDT1MAPTKDM4EL3MBTL1
SCHEMBL20866846 0.83 NUDT1 (0.52) TSHRNUDT1MAPTKDM4EL3MBTL1
SCHEMBL7365268 0.83 ALDH1A1 (0.66) TSHRNUDT1MAPTKDM4EL3MBTL1
SCHEMBL2544566 0.82 LMNA (0.68) NMT1NUDT1MAPTKDM4ENPSR1
SCHEMBL30639591 0.82 DHODH (0.55) TSHRMAPTKDM4EL3MBTL1GAA
SCHEMBL538115 0.81 NMT1 (0.61) TSHRNMT2NMT1MAPTKDM4E
SCHEMBL30647622 0.81 PTGS2 (0.53) NMT2NMT1NUDT1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023219456-A1 QUINOLINE-BASED HISTONE DEACETYLASE INHIBITORY SUBSTANCES, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION INCLUDING SAME AS ACTIVE INGREDIENT 숙명여자대학교 산학협력단 2023-11-16 WO disclosed