Phosphoric Acid

Phosphoric Acid

SCHEMBL3095605

Cc1cn([C@H]2CC[C@@H](C)O2)c(=O)[nH]c1=O.O=P(O)(O)O

nearest known ligand 0.64

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Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Phosphoric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TK1 P04183 6/20 0.52
TYMP P19971 2/20 0.48
DHFR P00374 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9549703 0.95 TK1 (0.50) TK1TYMPDHFR
SCHEMBL78118 0.93 TK1 (0.53) TK1DHFR
SCHEMBL19242604 0.93 TK1 (0.53) TK1DHFR
Pyrophosphoric Acid SCHEMBL1269545 0.93 POLB (0.54) TK1DHFR
SCHEMBL9549708 0.91 TK1 (0.48) TK1DHFR
Triphosphate SCHEMBL81707 0.91 POLB (0.55) TK1DHFR
SCHEMBL3154831 0.90 POLB (0.57) TK1DHFR
SCHEMBL9549653 0.88 TK1 (0.50) TK1DHFR
SCHEMBL9549656 0.87 TK1 (0.50) TK1DHFR
Phosphoric Acid SCHEMBL18249308 0.85 TK1 (0.58) TK1TYMP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115515968-A Allele-specific silencing of transforming growth factor beta-inducible genes with R124H mutation using short interfering RNA 阿维利诺美国实验室股份有限公司 2022-12-23 CN claimed
WO-2014031954-A1 HOMOPOLYMER MEDIATED NUCLEIC ACID AMPLIFICATION TUFTS UNIVERSITY (US) 2014-02-27 WO claimed
CN-115515968-A Allele-specific silencing of transforming growth factor beta-inducible genes with R124H mutation using short interfering RNA 阿维利诺美国实验室股份有限公司 2022-12-23 CN disclosed
US-9914950-B2 Homopolymer mediated nucleic acid amplification TUFTS UNIVERSITY (US) 2018-03-13 US disclosed
US-9340832-B2 Methods for enriching a variant nucleic acid from a nucleic acid population in a sample 360 GENOMICS LIMITED (GB) 2016-05-17 US disclosed
US-20150203887-A1 HOMOPOLYMER MEDIATED NUCLEIC ACID AMPLIFICATION TUFTS UNIVERSITY (US) 2015-07-23 US disclosed
WO-2014031954-A1 HOMOPOLYMER MEDIATED NUCLEIC ACID AMPLIFICATION TUFTS UNIVERSITY (US) 2014-02-27 WO disclosed
EP-2129797-B1 NUCLEIC ACID DETECTION OXITEC LTD (GB) 2013-04-03 EP disclosed
US-20100227320-A1 NUCLEIC ACID DETECTION 360 GENOMICS LIMITED (GB) 2010-09-09 US disclosed
EP-2129797-A2 NUCLEIC ACID DETECTION Oxitec Limited (GB) 2009-12-09 EP disclosed
WO-2008104794-A2 NUCLEIC ACID DETECTION OXITEC LIMITED (GB) 2008-09-04 WO disclosed
EP-1240355-B1 REMOVAL OF DYE-LABELED DIDEOXY TERMINATORS FROM DNA SEQUENCING REACTIONS CAMBREX BIO SCIENCE ROCKLAND I (US) 2008-08-27 EP disclosed
EP-1240355-A4 REMOVAL OF DYE-LABELED DIDEOXY TERMINATORS FROM DNA SEQUENCING REACTIONS PROLINX INC (US) 2004-12-08 EP disclosed
US-6818760-B1 COMPRISES ADSORBING UNINCORPORATED MOLECULES INTO POROUS HYDROPHOBIC PARTICLES ENCAPSULATED IN A HYDROPHILIC MATRIX; KITS PROLINX INCORPORATED 2004-11-16 US disclosed
EP-1240355-A1 REMOVAL OF DYE-LABELED DIDEOXY TERMINATORS FROM DNA SEQUENCING REACTIONS PROLINX, INC. (US) 2002-09-18 EP disclosed
US-6414136-B1 ADSORPTION OF FLUORESCENT DYE-LABELED MOLECULES NOT INCORPORATED IN POLYMER ONTO HYDROPHOBIC MATERIAL AFTER PASSING THROUGH HYDROPHILIC MATRIX PROLINX, INC. 2002-07-02 US disclosed
WO-2001025490-A1 REMOVAL OF DYE-LABELED DIDEOXY TERMINATORS FROM DNA SEQUENCING REACTIONS PROLINX, INC. (US) 2001-04-12 WO disclosed
WO-2001025491-A1 REMOVAL OF DYE-LABELED DIDEOXY TERMINATORS FROM DNA SEQUENCING REACTIONS PROLINX, INC. (US) 2001-04-12 WO disclosed
WO-1990014074-A1 IMPROVED LIPOSOMAL FORMULATIONS OF NUCLEOTIDES AND NUCLEOTIDE ANALOGUES VICAL, INC. (US) 1990-11-29 WO disclosed