SCHEMBL30965207

SCHEMBL30965207

O=C(O)CN1C(=O)c2cc(NS(=O)(=O)c3ccccc3)c(OOCCCCc3ccccc3)cc2C1=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.41
BCL2A1 Q16548 4/20 0.41
PTGDR2 Q9Y5Y4 5/20 0.39
MAPT P10636 2/20 0.38
METAP2 P50579 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
HDAC1 Q13547 2/20 0.37
AKR1B1 P15121 2/20 0.37
PTPN1 P18031 2/20 0.37
PTPN2 P17706 1/20 0.37
HTR6 P50406 1/20 0.37
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KMT2A Q03164 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30965221 0.91 MCL1 (0.40) MCL1BCL2A1PTGDR2METAP2HDAC1
SCHEMBL30965263 0.90 MCL1 (0.39) MCL1BCL2A1PTGDR2METAP2HDAC1
SCHEMBL30965245 0.84 MCL1 (0.38) MCL1BCL2A1PTGDR2MAPTCA12
SCHEMBL30965224 0.81 CYP19A1 (0.45) CA12CA9AKR1B1PTPN1PTPN2
SCHEMBL30965248 0.80 WDR5 (0.45) MAPTMETAP2CA12CA9ALDH1A1
SCHEMBL30965199 0.76 NAAA (0.36) MCL1BCL2A1PTGDR2KMT2A
SCHEMBL30965247 0.75 S1PR5 (0.38) MCL1BCL2A1ALDH1A1KMT2A
SCHEMBL30965174 0.75 AKR1B1 (0.42) CA12CA9AKR1B1PTPN1PTPN2
SCHEMBL30965268 0.73 ALDH1A1 (0.44) MAPTCA12CA9ALDH1A1NPSR1
SCHEMBL30965231 0.73 CA12 (0.47) MAPTCA12CA9AKR1B1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118125964-A Isoindoline-1, 3-diketone mPGES-1 inhibitor and application thereof 长江大学 2024-06-04 CN disclosed