SCHEMBL30965263

SCHEMBL30965263

O=C(O)CCCN1C(=O)c2cc(NS(=O)(=O)c3ccccc3)c(OOCCCCc3ccccc3)cc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.39
BCL2A1 Q16548 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 2/20 0.39
CYSLTR2 Q9NS75 1/20 0.39
CYSLTR1 Q9Y271 1/20 0.39
ACLY P53396 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
CASP1 P29466 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HDAC1 Q13547 1/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
NPC1 O15118 1/20 0.37
METAP2 P50579 1/20 0.37
S1PR5 Q9H228 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30965221 0.96 MCL1 (0.40) MCL1BCL2A1TDP1L3MBTL1RAB9A
SCHEMBL30965207 0.90 MCL1 (0.41) MCL1BCL2A1RAB9AKMT2AHDAC1
SCHEMBL30965247 0.85 S1PR5 (0.38) MCL1BCL2A1MAPK1CYSLTR2CYSLTR1
SCHEMBL30965250 0.82 RAB9A (0.45) TDP1L3MBTL1RAB9AMEN1KMT2A
SCHEMBL30965264 0.81 ACLY (0.44) MAPK1ACLYMEN1KMT2AGAA
SCHEMBL30965199 0.81 NAAA (0.36) MCL1BCL2A1CYSLTR2CYSLTR1ACLY
SCHEMBL30965151 0.77 CYP19A1 (0.44) TDP1L3MBTL1RAB9AS1PR5
SCHEMBL30965253 0.76 WDR5 (0.43) ACLYHSD17B10SMN1; SMN2METAP2S1PR5
SCHEMBL30965180 0.76 RAB9A (0.44) TDP1L3MBTL1RAB9AMEN1KMT2A
SCHEMBL30965193 0.74 MEN1 (0.52) TDP1L3MBTL1MAPK1RAB9ACYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118125964-A Isoindoline-1, 3-diketone mPGES-1 inhibitor and application thereof 长江大学 2024-06-04 CN disclosed