SCHEMBL3096956

SCHEMBL3096956

C1=COON=C1.NC(=O)NS(=O)(=O)c1ccccn1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.41
KAT6A Q92794 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
SLC40A1 Q9NP59 2/20 0.34
GLO1 Q04760 1/20 0.34
MMP2 P08253 2/20 0.34
PTGS2 P35354 5/20 0.34
METAP2 P50579 1/20 0.34
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
PKM P14618 1/20 0.33
RAB9A P51151 1/20 0.33
LGALS8 O00214 1/20 0.33
PTGS1 P23219 2/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
LOX P28300 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL729640 0.83 L3MBTL1 (0.50) NLRP3KAT6AL3MBTL1SLC40A1GLO1
SCHEMBL7959878 0.72 L3MBTL1 (0.51) NLRP3KAT6AL3MBTL1SLC40A1GLO1
SCHEMBL27771996 0.70 L3MBTL1 (0.49) NLRP3KAT6AL3MBTL1SLC40A1GLO1
SCHEMBL9370312 0.70 L3MBTL1 (0.49) NLRP3KAT6AL3MBTL1SLC40A1GLO1
SCHEMBL16549739 0.68 PKM (0.55) NLRP3KAT6AL3MBTL1SLC40A1GLO1
SCHEMBL25294544 0.66 P4HTM (0.56) NLRP3KAT6AL3MBTL1PTGS2NPC1
SCHEMBL18157894 0.66 PTGS2 (0.71) NLRP3L3MBTL1PTGS2METAP2NPC1
SCHEMBL136276 0.65 MEN1 (0.40) L3MBTL1MMP2PTGS2PKMPTGS1
SCHEMBL2059520 0.65 MKNK1 (0.31)
SCHEMBL10430944 0.65 NLRP3 (0.47) NLRP3KAT6AL3MBTL1SLC40A1GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100190992-A1 Nicotinamide derivatives as synthesis units for producing agrochemical substances, and method for the production thereof BAYER CROPSCIENCE AG (DE) 2010-07-29 US disclosed
US-20100184973-A1 Method for producing dioxazine derivatives BAYER CROPSCIENCE AG (DE) 2010-07-22 US disclosed
CN-101687804-A Method for producing dioxazine derivatives BAYER CROPSCIENCE AG 2010-03-31 CN disclosed
CN-101679398-A Nicotinamide derivatives useful as synthetic units for the preparation of agricultural chemicals, and process for the preparation thereof BAYER CROPSCIENCE AG 2010-03-24 CN disclosed
EP-2160391-A1 NICOTINAMIDE DERIVATIVES AS SYNTHESIS UNITS FOR PRODUCING AGROCHEMICAL SUBSTANCES, AND METHOD FOR THE PRODUCTION THEREOF Bayer CropScience AG (DE) 2010-03-10 EP disclosed
CN-101558036-A Process for preparing 2-aminooxyethanol BAYER CROPSCIENCE AG (DE) 2009-10-14 CN disclosed
WO-2008155003-A1 NICOTINAMIDE DERIVATIVES AS SYNTHESIS UNITS FOR PRODUCING AGROCHEMICAL SUBSTANCES, AND METHOD FOR THE PRODUCTION THEREOF BAYER CROPSCIENCE AG (DE) 2008-12-24 WO disclosed
EP-1728430-A1 Herbicidal agents Bayer CropScience GmbH (DE) 2006-12-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100190992-A1 Nicotinamide derivatives as synthesis units for producing agrochemical substances, and method for the production thereof NAMPT, NQO1, NNT NLRP3 1255/4885KAT6A 4551/4885L3MBTL1 4513/4885
US-20100184973-A1 Method for producing dioxazine derivatives CYP4Z1, CYP1A1, CYP2F1 NLRP3 1724/4885KAT6A 3520/4885L3MBTL1 4848/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.