SCHEMBL3137112

SCHEMBL3137112

CNC1(COc2cncc(-c3cccc(C#N)c3)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 3/20 0.44
GABRB3 P28472 3/20 0.44
GABRA5 P31644 3/20 0.44
GABRA3 P34903 3/20 0.44
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
CHRNB2 P17787 2/20 0.40
NEK1 Q96PY6 1/20 0.40
CHRNA4 P43681 1/20 0.40
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
CHRNB1 P11230 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNB3 Q05901 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3772099 0.99 GABRG2 (0.46) GABRG2GABRB3GABRA5GABRA3CYP11B1
SCHEMBL3150657 0.87 CYP11B1 (0.43) CYP11B1CYP11B2CHRNB2CHRNA4PRMT5
Hydrochloric Acid SCHEMBL3781163 0.86 CYP11B1 (0.42) CYP11B1CYP11B2CHRNB2CHRNA4PRMT5
SCHEMBL3150645 0.84 CYP11B1 (0.47) CYP11B1CYP11B2
SCHEMBL3142735 0.84 S1PR1 (0.38) CYP11B1CYP11B2CHRNB2CHRNA4CHRNB1
SCHEMBL3147229 0.83 CHRNB2 (0.49) CYP11B1CYP11B2CHRNB2CHRNA4CHRNB1
SCHEMBL3147306 0.83 INPPL1 (0.43) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3
Hydrochloric Acid SCHEMBL3141660 0.83 CYP11B1 (0.46) CYP11B1CYP11B2
SCHEMBL3137054 0.83 CYP11B2 (0.39) CYP11B1CYP11B2CHRNB2CHRNA4PRMT5
SCHEMBL3146014 0.83 CHRNB1 (0.52) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed