Pyridine

Pyridine

SCHEMBL3147614

O=S(=O)(O)OOO.c1ccncc1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 2/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CA2 P00918 1/20 0.39
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridine SCHEMBL28257184 0.88 CA2 (0.53) NAPRTTSHRTDP1CA2MAPT
Pyridine SCHEMBL2424842 0.88 CA2 (0.53) NAPRTTSHRTDP1CA2MAPT
Pyridine SCHEMBL28040883 0.86 CA2 (0.50) NAPRTTSHRTDP1CA2
Pyridine SCHEMBL8570319 0.84 NAPRT (0.43) NAPRTTSHRTDP1CA2
Pyridine SCHEMBL5606559 0.84 NAPRT (0.43) NAPRTTSHRTDP1CA2
Pyridine SCHEMBL6671998 0.80 NAPRT (0.39) NAPRTTSHRTDP1CA2
Pyridine SCHEMBL9785253 0.78 NAPRT (0.47) NAPRTTSHRTDP1CA2MAPT
Pyridine SCHEMBL2255454 0.78 NAPRT (0.47) NAPRTTSHRTDP1CA2MAPT
Pyridine SCHEMBL984983 0.78 TSHR (0.53) NAPRTTSHRTDP1
Pyridine SCHEMBL407438 0.77 NAPRT (0.60) NAPRTTSHRTDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110294748-A A kind of synthetic method for Ge Lieting key intermediate 浙江沙星科技有限公司 2019-10-01 CN claimed
CN-109803952-A Sulfamic acid derivatives and preparation method thereof 魁北克电力公司 2019-05-24 CN claimed
CN-108349938-A Salts of Pim Kinase Inhibitors 因赛特公司 2018-07-31 CN claimed
CN-107501359-A A kind of Fondaparinux sodium impurity compound and preparation method and application 深圳市海滨制药有限公司 2017-12-22 CN claimed
EP-1304338-B1 Process for the preparation of Chondroitin sulfates from K4 Polysaccharide and obtained products IBSA INST BIOCHIMIQUE SA (CH) 2008-08-13 EP claimed
US-20030100534-A1 Process for the preparation of chondroitin sulfates from K4 polysaccharide and obtained products IBSA INSTITUT BIOCHIMIQUE S.A. (CH) 2003-05-29 US claimed
EP-1304338-A1 Process for the preparation of Chondroitin sulfates from K4 Polysaccharide and obtained products Ibsa Institut Biochimique S.A. (CH) 2003-04-23 EP claimed
CN-110218213-A The thick cyclics of pyrans, preparation method and use 北京天一绿甫医药科技有限公司 2019-09-10 CN disclosed
CN-106029057-B Oral formulations of pyrrolidine derivatives 奥布赛瓦股份公司 2019-09-03 CN disclosed
CN-110121499-A (aza) indole-, benzothiophene-and benzofuran-3-sulfonamides 优时比制药有限公司 2019-08-13 CN disclosed
CN-109928905-A As oxytocins/pitressin V1a receptor antagonist pyrrolidin derivatives 奥布赛瓦股份公司 2019-06-25 CN disclosed
CN-109937206-A Polymerizable compound, and method for producing borane phosphate oligomer 学校法人东京理科大学 2019-06-25 CN disclosed
CN-109879979-A A kind of antioxidant and preparation method thereof 武汉轻工大学 2019-06-14 CN disclosed
US-20030060448-A1 Use of hyaluronic acid derivatives in the preparation of biomaterials with a physical haemostatic and plugging activity and a preventive activity in the formation of adhesions following anastomosis ANIKA THERAPEUTICS S.R.L. (IT) 2003-03-27 US disclosed
EP-0971961-B1 N-SULPHATED HYALURONIC ACID COMPOUNDS, DERIVATIVES THEREOF AND A PROCESS FOR THEIR PREPARATION FIDIA ADVANCED BIOPOLYMERS SRL (IT) 2002-12-04 EP disclosed
US-20020037874-A1 N-sulphated hyaluronic acid compounds, derivatives thereof and a process for their preparation FIDIA ADVANCED BIOPOLYMERS 2002-03-28 US disclosed
EP-0999859-A2 USE OF HYALURONIC ACID DERIVATIVES IN THE PREPARATION OF BIOMATERIALS FIDIA ADVANCED BIOPOLYMERS S.R.L. (IT) 2000-05-17 EP disclosed
WO-1999004828-A2 USE OF HYALURONIC ACID DERIVATIVES IN THE PREPARATION OF BIOMATERIALS FIDIA ADVANCED BIOPOLYMERS, S.R.L. (IT) 1999-02-04 WO disclosed
EP-0439555-A1 NOVEL DERMATAN SULFATE AND HEPARIN OLIGOSACCHARIDES HAVING ANTIATHEROSCLEROTIC ACTIVITY. OPOCRIN SPA (IT) 1991-08-07 EP disclosed
WO-1990004607-A2 NOVEL DERMATAN SULFATE AND HEPARIN OLIGOSACCHARIDES HAVING ANTIATHEROSCLEROTIC ACTIVITY OPOCRIN S.P.A. LABORATORIO FARMACOBIOLOGICO (IT) 1990-05-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030100534-A1 Process for the preparation of chondroitin sulfates from K4 polysaccharide and obtained products CSGALNACT1, DDOST, STT3B NAPRT 803/4885TSHR 4098/4885TDP1 4431/4885
US-20020037874-A1 N-sulphated hyaluronic acid compounds, derivatives thereof and a process for their preparation HPSE, CD44, HEXD NAPRT 110/4885TSHR 3434/4885TDP1 4196/4885
US-20030060448-A1 Use of hyaluronic acid derivatives in the preparation of biomaterials with a physical haemostatic and plugging activity and a preventive activity in the formation of adhesions following anastomosis MMP1, PLG, CD44 NAPRT 2185/4885TSHR 4025/4885TDP1 2801/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.