Daunorubicin

Daunorubicin

SCHEMBL319903

COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(C)=O)C[C@@H]3O[C@@H]1C[C@H](N)[C@H](O)[C@H](C)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TOP2A

The experimentally established mechanism targets of Daunorubicin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A known ✓ P11388 5/20 1.00
MEN1 O00255 10/20 1.00
THRB P10828 10/20 1.00
KMT2A Q03164 10/20 1.00
BLM P54132 9/20 1.00
RECQL P46063 8/20 1.00
BRCA1 P38398 7/20 1.00
SMN1; SMN2 Q16637 7/20 1.00
HIF1A Q16665 7/20 1.00
MAPT P10636 7/20 1.00
TDP1 Q9NUW8 6/20 1.00
MAPK1 P28482 6/20 1.00
CYP3A4 P08684 5/20 1.00
USP2 O75604 5/20 1.00
HTT P42858 5/20 1.00
CYP1A2 P05177 4/20 1.00
CHRM1 P11229 4/20 1.00
KDM4E B2RXH2 4/20 1.00
ALDH1A1 P00352 4/20 1.00
TP53 P04637 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Daunorubicin SCHEMBL6423269 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL15159339 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL6423273 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL12864552 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL289431 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL24914323 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL18926545 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL13840952 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL22694307 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL10061862 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114650823-A Pharmaceutical composition comprising FLT3 inhibitor and chemotherapeutic agent for the treatment of acute myeloid leukemia 韩美药品株式会社 2022-06-21 CN claimed
US-12350265-B2 Pharmaceutical composition for treating acute myeloid leukemia, containing FLT3 inhibitor and chemotherapeutic agents HANMI PHARM. CO., LTD. (KR) 2025-07-08 US disclosed
US-12295957-B2 Ascorbic acid and quinone compounds in combination with an antiparasitic agent for treating a parasitic disease IC-MedTech Corp. (US) 2025-05-13 US disclosed
US-20240398755-A1 ASCORBIC ACID AND QUINONE COMPOUNDS FOR TREATING CHAGAS DISEASE IC-MedTech Corp. 2024-12-05 US disclosed
US-11998523-B2 Ascorbic acid and quinone compounds for treating Chagas disease IC-MedTech Corp. (US) 2024-06-04 US disclosed
US-20240165084-A1 ASCORBIC ACID AND QUINONE COMPOUNDS IN COMBINATION WITH AN ANTIPARASITIC AGENT FOR TREATING A PARASITIC DISEASE IC-MedTech Corp. 2024-05-23 US disclosed
US-11872233-B2 Ascorbic acid and quinone compounds in combination with an antiparasitic agent for treating a parasitic disease IC-MedTech Corp. (US) 2024-01-16 US disclosed
US-20230364086-A1 COMBINATION THERAPIES WITH EHMT2 INHIBITORS Epizyme, Inc. 2023-11-16 US disclosed
US-11672800-B2 Combination therapies with EHMT2 inhibitors Epizyme, Inc. (US) 2023-06-13 US disclosed
US-20220409577-A1 INTRATUMORAL ADMINISTRATION OF ASCORBIC ACID AND QUINONE COMPOUNDS FOR TUMOR TREATMENT IC-MedTech Corp. 2022-12-29 US disclosed
US-9737614-B2 Fucoidan nanogels and methods of their use and manufacture MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2017-08-22 US disclosed
US-20160193349-A1 FUCOIDAN NANOGELS AND METHODS OF THEIR USE AND MANUFACTURE NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-07-07 US disclosed
US-20150328254-A1 FUCOIDAN NANOGELS AND METHODS OF THEIR USE AND MANUFACTURE MEMORIAL SLOAN KETTERING CANCER CENTER 2015-11-19 US disclosed
US-8092828-B2 Administering mixture of cytarabine and anthracycline CELATOR PHARMACEUTICALS, INC. (US) 2012-01-10 US disclosed
US-20100303895-A1 FIXED DRUG RATIOS FOR TREATMENT OF HEMATOPOIETIC CANCERS AND PROLIFERATIVE DISORDERS CELATOR PHARMACEUTICALS, INC. 2010-12-02 US disclosed
WO-2010133700-A1 PHARMACEUTICAL COMPOSITION COMPRISING MICROBUBBLES FOR TARGETED TUMOR THERAPY LUDWIG-MAXIMILIANS-UNIVERSITÄT MÜNCHEN (DE) 2010-11-25 WO disclosed
EP-2253308-A1 Pharmaceutical composition comprising microbubbles for targeted tumor therapy Ludwig-Maximilians-Universität München (DE) 2010-11-24 EP disclosed
EP-2120568-A2 FIXED DRUG RATIOS FOR TREATMENT OF HEMATOPOIETIC CANCERS AND PROLIFERATIVE DISORDERS Celator Pharmaceuticals, Inc. (US) 2009-11-25 EP disclosed
US-20080199515-A1 FIXED DRUG RATIOS FOR TREATMENT OF HEMATOPOIETIC CANCERS AND PROLIFERATIVE DISORDERS Jazz Pharmaceuticals Therapeutics, Inc. 2008-08-21 US disclosed
WO-2008101214-A2 FIXED DRUG RATIOS FOR TREATMENT OF HEMATOPOIETIC CANCERS AND PROLIFERATIVE DISORDERS CELATOR PHARMACEUTICALS, INC. (US) 2008-08-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230364086-A1 COMBINATION THERAPIES WITH EHMT2 INHIBITORS EHMT2, BHMT, SHMT2 TOP2A 199/4885MEN1 1229/4885THRB 916/4885
US-11872233-B2 Ascorbic acid and quinone compounds in combination with an antiparasitic agent for treating a parasitic disease NQO1, ADH7, CYP27B1 TOP2A 2184/4885MEN1 2407/4885THRB 3967/4885
US-12350265-B2 Pharmaceutical composition for treating acute myeloid leukemia, containing FLT3 inhibitor and chemotherapeutic agents FLT3, MCL1, CSF3R TOP2A 2835/4885MEN1 1801/4885THRB 2992/4885
US-20220409577-A1 INTRATUMORAL ADMINISTRATION OF ASCORBIC ACID AND QUINONE COMPOUNDS FOR TUMOR TREATMENT NDUFB7, NDUFA12, NDUFB11 TOP2A 859/4885MEN1 1050/4885THRB 2730/4885
US-20240165084-A1 ASCORBIC ACID AND QUINONE COMPOUNDS IN COMBINATION WITH AN ANTIPARASITIC AGENT FOR TREATING A PARASITIC DISEASE NQO1, ADH7, CYP27B1 TOP2A 2184/4885MEN1 2407/4885THRB 3967/4885
US-11998523-B2 Ascorbic acid and quinone compounds for treating Chagas disease NQO1, ADH7, TALDO1 TOP2A 2041/4885MEN1 2264/4885THRB 3280/4885
US-12295957-B2 Ascorbic acid and quinone compounds in combination with an antiparasitic agent for treating a parasitic disease NQO1, ADH7, CYP27B1 TOP2A 2184/4885MEN1 2407/4885THRB 3967/4885
US-11672800-B2 Combination therapies with EHMT2 inhibitors EHMT2, BHMT, SHMT2 TOP2A 199/4885MEN1 1229/4885THRB 916/4885
US-20240398755-A1 ASCORBIC ACID AND QUINONE COMPOUNDS FOR TREATING CHAGAS DISEASE NQO1, ADH7, TALDO1 TOP2A 2041/4885MEN1 2264/4885THRB 3280/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.