Acetic Acid

Acetic Acid

SCHEMBL3212866

CC(=O)O.COc1cccc(OC)c1CN1Cc2ccc(-c3cccnc3)cc2N=C1N

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 3/20 0.44
MKNK2 Q9HBH9 3/20 0.44
HCRTR1 O43613 4/20 0.41
HCRTR2 O43614 4/20 0.41
F2 P00734 1/20 0.38
F12 P00748 1/20 0.38
POLB P06746 1/20 0.38
CYP11B2 P19099 3/20 0.38
CYP11B1 P15538 2/20 0.38
BACE1 P56817 4/20 0.38
CTSD P07339 3/20 0.38
BACE2 Q9Y5Z0 3/20 0.38
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CREBBP Q92793 1/20 0.37
MAPK1 P28482 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4716955 0.94 HCRTR1 (0.42) MKNK1MKNK2HCRTR1HCRTR2CYP11B2
Acetic Acid SCHEMBL3263693 0.91 CTSD (0.44) HCRTR1HCRTR2BACE1CTSDMEN1
Acetic Acid SCHEMBL3206340 0.87 CTSD (0.39) BACE1CTSDSMN1; SMN2
SCHEMBL4715532 0.86 CTSD (0.48) HCRTR1HCRTR2BACE1CTSD
Acetic Acid SCHEMBL3207125 0.83 CTSD (0.39) BACE1CTSDMEN1LMNAKMT2A
SCHEMBL4718491 0.81 CTSD (0.40) BACE1CTSDABL1BCR
Acetic Acid SCHEMBL3216929 0.81 SIGMAR1 (0.42) BACE1CTSDBACE2MEN1KMT2A
Acetic Acid SCHEMBL3222963 0.79 HIF1A (0.38) BACE1CTSDMEN1KMT2AMAPK1
SCHEMBL4719286 0.76 CTSD (0.43) CTSDMEN1LMNAKMT2ASMN1; SMN2
SCHEMBL4716520 0.76 GRIN2B (0.42) HCRTR1HCRTR2BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140221371-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS AbbVie Deutschland GmbH & Co. KG (DE) 2014-08-07 US disclosed
US-20100041698-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS ABBVIE DEUTSCHLAND GMBH & CO KG (DE) 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221371-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS HTR5A, HTR1A, HTR2C MKNK1 1366/4885MKNK2 1225/4885HCRTR1 110/4885
US-20100041698-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS HTR5A, HTR1A, HTR2C MKNK1 1366/4885MKNK2 1225/4885HCRTR1 110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.