SCHEMBL3223963

SCHEMBL3223963

Cc1cc(S(=O)(=O)F)ccc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
TDP1 Q9NUW8 4/20 0.47
CYP3A4 P08684 4/20 0.47
TSHR P16473 3/20 0.46
S100B P04271 1/20 0.46
LMNA P02545 1/20 0.45
CA12 O43570 4/20 0.44
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA4 P22748 4/20 0.44
CA6 P23280 4/20 0.44
CA5A P35218 4/20 0.44
CA7 P43166 4/20 0.44
CA9 Q16790 4/20 0.44
CA14 Q9ULX7 4/20 0.44
CA5B Q9Y2D0 4/20 0.44
G6PD P11413 1/20 0.40
IDE P14735 1/20 0.40
THRB P10828 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7997480 0.83 ALDH1A1 (0.46) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL436337 0.83 ALDH1A1 (0.55) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL31120743 0.81 TDP1 (0.69) ALDH1A1TDP1CYP3A4TSHRS100B
SCHEMBL878966 0.81 CA2 (0.67) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL30291216 0.81 CA2 (0.67) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL1365469 0.81 TDP1 (0.69) ALDH1A1TDP1CYP3A4TSHRS100B
SCHEMBL4639254 0.81 G6PD (0.60) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL10391068 0.80 ALDH1A1 (0.61) ALDH1A1TDP1CYP3A4TSHRCA12
SCHEMBL10412670 0.80 LMNA (0.61) ALDH1A1TDP1TSHRLMNAPKM
SCHEMBL5623940 0.80 ALDH1A1 (0.60) ALDH1A1TDP1CYP3A4TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8329755-B2 Methods for treating retroviral infections ROCHE PALO ALTO LLC (US) 2012-12-11 US disclosed
US-8329755-B2 Methods for treating retroviral infections ROCHE PALO ALTO LLC (US) 2012-12-11 US disclosed
CN-1946680-B Non-nucleoside reverse transcriptase inhibitors F. HOFFMANN-LA ROCHE AG (CH) 2011-04-06 CN disclosed
US-20100041648-A1 METHODS FOR TREATING RETROVIRAL INFECTIONS DUNN JAMES PATRICK 2010-02-18 US disclosed
US-20100041648-A1 METHODS FOR TREATING RETROVIRAL INFECTIONS DUNN JAMES PATRICK 2010-02-18 US disclosed
US-7625949-B2 Methods for treating retroviral infections ROCHE PALO ALTO LLC (US) 2009-12-01 US disclosed
US-7625949-B2 Methods for treating retroviral infections ROCHE PALO ALTO LLC (US) 2009-12-01 US disclosed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed
CN-1946680-A Non-nucleoside reverse transcriptase inhibitors HOFFMANN LA ROCHE (CH) 2007-04-11 CN disclosed
US-7166738-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-01-23 US disclosed
US-7166738-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-01-23 US disclosed
US-7166738-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-01-23 US disclosed
EP-1742908-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-01-17 EP disclosed
WO-2005102989-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-11-03 WO disclosed
US-20050239881-A1 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC 2005-10-27 US disclosed
US-20050239880-A1 Methods for treating retroviral infections ROCHE PALO ALTO LLC 2005-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041648-A1 METHODS FOR TREATING RETROVIRAL INFECTIONS CCR5, CXCR4, CCR1 ALDH1A1 261/4885TDP1 3239/4885CYP3A4 3060/4885
US-20050239880-A1 Methods for treating retroviral infections CCR5, CD38, CD4 ALDH1A1 428/4885TDP1 3293/4885CYP3A4 2749/4885
US-20050239881-A1 Non-nucleoside reverse transcriptase inhibitors RPP30, PNP, RTF1 ALDH1A1 2794/4885TDP1 688/4885CYP3A4 2342/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.