SCHEMBL3240923

SCHEMBL3240923

CC(C)(C)OC(=O)CN1C(=O)CCc2cc(-c3cc(Cl)cc(Cl)c3)cnc21

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.38
CYP11B2 P19099 6/20 0.38
MAPK1 P28482 3/20 0.36
CCKBR P32239 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
BMPR1B O00238 1/20 0.33
BMPR1A P36894 1/20 0.33
ACVRL1 P37023 1/20 0.33
ACVR1 Q04771 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3240957 0.86 GRIN2B (0.41) METMAPK1
SCHEMBL3241068 0.84 CYP11B2 (0.41) CYP11B2BMPR1BBMPR1AACVRL1ACVR1
SCHEMBL3245592 0.82 ALDH1A1 (0.37) METMAPK1CCKBRKDM4EALDH1A1
SCHEMBL13521571 0.81 USP2 (0.42) MAPK1KDM4EALDH1A1
SCHEMBL3246493 0.77 FNTA (0.39) CYP11B2MAPK1KDM4EALDH1A1
SCHEMBL3246489 0.76 CYP11B2 (0.36) CYP11B2KDM4EALDH1A1BMPR1BBMPR1A
SCHEMBL3128762 0.75 SMN1; SMN2 (0.42) CYP11B2MAPK1KDM4EALDH1A1
SCHEMBL3130951 0.73 ESR1 (0.43) CYP11B2MAPK1KDM4EALDH1A1
SCHEMBL3118590 0.73 ESR2 (0.45) CYP11B2MAPK1KDM4EALDH1A1
SCHEMBL9532098 0.71 PLA2G10 (0.40) CCKBRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed