SCHEMBL3301765

SCHEMBL3301765

COC(=O)N1CC2CCC(=O)CC2CC1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
MMP2 P08253 4/20 0.33
ANPEP P15144 3/20 0.33
ATM Q13315 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8983770 1.00 TSHR (0.36) TSHRMMP2ANPEPATMMEN1
SCHEMBL6798706 1.00 TSHR (0.36) TSHRMMP2ANPEPATMMEN1
SCHEMBL3307394 1.00 TSHR (0.36) TSHRMMP2ANPEPATMMEN1
SCHEMBL8866598 0.90 MMP2 (0.39) TSHRMMP2ANPEP
SCHEMBL8867224 0.90 MMP2 (0.39) TSHRMMP2ANPEP
SCHEMBL13390232 0.89 TSHR (0.36) TSHRMMP2ANPEPTHRB
SCHEMBL3304315 0.87 HSD17B10 (0.38)
SCHEMBL3301971 0.87 HSD17B10 (0.38)
SCHEMBL6607994 0.86 AGTR2 (0.35) TSHRMEN1KMT2A
SCHEMBL25475425 0.84 ALDH1A1 (0.32) TSHRMMP2ANPEPKMT2ATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250074887-A1 PHARMACEUTICAL COMPOSITIONS OF 6-(2-(2H-TETRAZOL-5-YL)ETHYL)DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID AND DERIVATIVES THEREOF Sea Pharmaceuticals LLC. (US) 2025-03-06 US disclosed
US-20100094014-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS MARTINEZ-PEREZ JOSE ANTONIO 2010-04-15 US disclosed
EP-2166003-A1 Excitatory amino acid receptor antagonists Eli Lilly & Company (US) 2010-03-24 EP disclosed
US-7601738-B2 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 2009-10-13 US disclosed
EP-1368032-B1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-11 EP disclosed
US-7205313-B2 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 2007-04-17 US disclosed
US-20060100237-A1 Excitatory amino acid receptor antagonists ARNOLD MACKLIN B 2006-05-11 US disclosed
US-6953805-B2 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 2005-10-11 US disclosed
US-20050170999-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS FILLA SANDRA A (US) 2005-08-04 US disclosed
US-6924294-B2 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 2005-08-02 US disclosed
US-5670516-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1997-09-23 US disclosed
US-5648492-A Process for preparing isoquinoline compounds ELI LILLY AND COMPANY (US) 1997-07-15 US disclosed
US-5637712-A CATALYTIC HYDROGENNATION ELI LILLY AND COMPANY (US) 1997-06-10 US disclosed
US-5606062-A STEREOSELECTIVE REDUCTION ELI LILLY AND COMPANY (US) 1997-02-25 US disclosed
US-5527810-A USEFUL IN THE TREATMENT OF NEUROLOGICAL DISORDERS ELI LILLY AND COMPANY (US) 1996-06-18 US disclosed
US-5446051-A Nervous system disorder and brain disorder ELI LILLY AND COMPANY (US) 1995-08-29 US disclosed
US-5399696-A Excitatory amino acid receptor antagonists; nervous system disorders ELI LILLY AND COMPANY (US) 1995-03-21 US disclosed
US-5356902-A Central nervous system disorders ELI LILLY AND COMPANY (US) 1994-10-18 US disclosed
EP-0590789-A1 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 1994-04-06 EP disclosed
US-5284957-A Substituted 1H- or 2H-tetrazoles ELI LILLY AND COMPANY (US) 1994-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250074887-A1 PHARMACEUTICAL COMPOSITIONS OF 6-(2-(2H-TETRAZOL-5-YL)ETHYL)DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID AND DERIVATIVES THEREOF GABRQ, GRIK5, CYP3A7 TSHR 3434/4885MMP2 2337/4885ANPEP 2525/4885
US-20100094014-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS SLC1A2, SLC1A1, GRIN1 TSHR 642/4885MMP2 4471/4885ANPEP 668/4885
US-20050170999-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS SLC1A2, SLC1A1, SLC1A3 TSHR 807/4885MMP2 4107/4885ANPEP 787/4885
US-20060100237-A1 Excitatory amino acid receptor antagonists SLC1A2, SLC1A1, GRIN1 TSHR 642/4885MMP2 4471/4885ANPEP 668/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.