SCHEMBL3353261

SCHEMBL3353261

CC[C@H](NC(=O)[C@@H]1CNC[C@H]1c1cc(Cl)cc(Cl)c1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
REN P00797 5/20 0.44
KCNQ3 O43525 3/20 0.42
KCNQ2 O43526 3/20 0.42
KCNQ4 P56696 1/20 0.41
KCNQ5 Q9NR82 1/20 0.41
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ROCK2 O75116 2/20 0.39
EPHX2 P34913 2/20 0.39
CMA1 P23946 1/20 0.39
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3416539 0.87 GPR88 (0.45) GPR88TDP1TAS1R3TAS1R1REN
SCHEMBL3353138 0.85 KCNQ3 (0.52) KCNQ3KCNQ2KCNQ4KCNQ5LMNA
SCHEMBL3346531 0.82 GPR88 (0.66) GPR88TDP1KCNQ3KCNQ2
SCHEMBL3353012 0.81 KCNH2 (0.59) GPR88TDP1KCNQ3KCNQ2KCNQ4
SCHEMBL3353295 0.79 GPR88 (0.52) GPR88TDP1KCNQ3KCNQ2
SCHEMBL3346676 0.77 KCNQ3 (0.53) KCNQ3KCNQ2KCNQ4KCNQ5ROCK2
SCHEMBL3353133 0.77 KCNH2 (0.47) RENKCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL3346539 0.75 KCNH2 (0.57) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL3353142 0.75 MC4R (0.62) ALDH1A1HPGDHSD17B10MAPTNPSR1
SCHEMBL3346373 0.75 KCNH2 (0.57) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed