SCHEMBL3353295

SCHEMBL3353295

CC[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(OC(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 2/20 0.52
PDE2A O00408 10/20 0.47
KCNH2 Q12809 4/20 0.45
PDE5A O76074 1/20 0.42
PDE1A P54750 1/20 0.42
PDE3A Q14432 1/20 0.42
GPR139 Q6DWJ6 1/20 0.42
KCNQ3 O43525 1/20 0.41
KCNQ2 O43526 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346531 0.88 GPR88 (0.66) GPR88KCNH2KCNQ3KCNQ2TDP1
SCHEMBL3353031 0.87 KCNH2 (0.59) PDE2AKCNH2GPR139KCNQ3KCNQ2
SCHEMBL3353012 0.87 KCNH2 (0.59) GPR88KCNH2KCNQ3KCNQ2TDP1
SCHEMBL3346914 0.79 KCNH2 (0.52) PDE2AKCNH2GPR139KCNQ3KCNQ2
SCHEMBL3416539 0.79 GPR88 (0.45) GPR88KCNH2KCNQ3KCNQ2TDP1
SCHEMBL3353261 0.79 GPR88 (0.46) GPR88KCNQ3KCNQ2TDP1
SCHEMBL3348200 0.78 KCNH2 (0.52) KCNH2GPR139
SCHEMBL3353035 0.78 MC4R (0.56) KCNH2
SCHEMBL17230469 0.74 GPR88 (0.66) GPR88KCNQ3KCNQ2
SCHEMBL3412005 0.74 KCNH2 (0.55) GPR88KCNH2KCNQ3KCNQ2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed