SCHEMBL335834

SCHEMBL335834

Nc1nc2ccc(NC(=O)C(O)C(NC(=O)c3ccc4ccccc4n3)c3ccccc3)cc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
NFKB1 P19838 2/20 0.42
NFKB2 Q00653 2/20 0.42
RELA Q04206 2/20 0.42
ACP1 P24666 1/20 0.41
HDAC1 Q13547 2/20 0.40
ALDH1A1 P00352 4/20 0.40
NPC1 O15118 3/20 0.40
MAPT P10636 2/20 0.39
POLB P06746 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ABL1 P00519 1/20 0.39
FABP6 P51161 1/20 0.39
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CCR1 P32246 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL336443 0.89 SMN1; SMN2 (0.43) RAB9ASMN1; SMN2ACP1NPC1MAPT
SCHEMBL335390 0.86 ABL1 (0.44) RAB9ASMN1; SMN2ACP1ALDH1A1NPC1
SCHEMBL15282212 0.86 ACP1 (0.46) RAB9ASMN1; SMN2ACP1ALDH1A1NPC1
SCHEMBL15282285 0.86 ACP1 (0.46) RAB9ASMN1; SMN2ACP1ALDH1A1NPC1
SCHEMBL335316 0.85 ALOX15 (0.41)
SCHEMBL335351 0.85 EGFR (0.50) RAB9ASMN1; SMN2ACP1HDAC1ALDH1A1
SCHEMBL336367 0.84 MAPT (0.47) RAB9ASMN1; SMN2ACP1ALDH1A1NPC1
SCHEMBL335948 0.84 ABL1 (0.45) RAB9ASMN1; SMN2ACP1HDAC1ALDH1A1
SCHEMBL335570 0.83 PIN1 (0.47) RAB9AACP1HDAC1MAPTABL1
SCHEMBL335878 0.82 ABL1 (0.43) SMN1; SMN2ACP1HDAC1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097758-B2 Isoserine derivatives for use as coagulation factor IXa inhibitors SANOFI-AVENTIS (FR) 2012-01-17 US claimed