SCHEMBL336443

SCHEMBL336443

Nc1nc2ccc(NC(=O)C(O)C(NC(=O)c3cnc4ccccc4n3)c3ccccc3)cc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.43
NPC1 O15118 2/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
GAA P10253 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ACP1 P24666 1/20 0.40
SIRT1 Q96EB6 1/20 0.39
AKR1B1 P15121 2/20 0.39
GRN P28799 1/20 0.39
SORT1 Q99523 1/20 0.39
ABL1 P00519 1/20 0.39
FABP6 P51161 1/20 0.39
CCR1 P32246 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL335834 0.89 RAB9A (0.42) SMN1; SMN2NPC1MAPTRAB9AGAA
SCHEMBL15282285 0.85 ACP1 (0.46) SMN1; SMN2NPC1MAPTRAB9AGAA
SCHEMBL15282212 0.85 ACP1 (0.46) SMN1; SMN2NPC1MAPTRAB9AGAA
SCHEMBL335316 0.84 ALOX15 (0.41)
SCHEMBL336367 0.84 MAPT (0.47) SMN1; SMN2NPC1MAPTRAB9AKDM4E
SCHEMBL335948 0.83 ABL1 (0.45) SMN1; SMN2NPC1MAPTRAB9AKDM4E
SCHEMBL335570 0.82 PIN1 (0.47) MAPTRAB9AACP1ABL1FABP6
SCHEMBL335351 0.82 EGFR (0.50) SMN1; SMN2NPC1RAB9AGAAKDM4E
SCHEMBL335390 0.82 ABL1 (0.44) SMN1; SMN2NPC1MAPTRAB9AKDM4E
SCHEMBL335729 0.82 F7 (0.43) ACP1ABL1FABP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097758-B2 Isoserine derivatives for use as coagulation factor IXa inhibitors SANOFI-AVENTIS (FR) 2012-01-17 US claimed