Fluprostenol

Fluprostenol

SCHEMBL3364535

O=C(O)CCCC=CC[C@@H]1[C@@H](C=CC(O)COc2cccc(C(F)(F)F)c2)[C@H](O)C[C@@H]1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGFR P43088 16/20 1.00
PTGER3 P43115 5/20 1.00
ABCC4 O15439 2/20 0.81
ABCB11 O95342 1/20 0.81
TBXA2R P21731 3/20 0.78
PTGER1 P34995 2/20 0.78
THRB P10828 1/20 0.78
PTGER2 P43116 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluprostenol SCHEMBL16414486 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL16414497 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL2744986 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL10015915 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL24342036 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL13260302 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL24342073 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL6750653 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL230607 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R
Fluprostenol SCHEMBL20860290 1.00 PTGFR (1.00) PTGFRPTGER3ABCC4ABCB11TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100105771-A1 AMINO ACID SALTS OF PROSTAGLANDINS NOVAER HOLDINGS, INC. 2010-04-29 US claimed
US-20250074935-A1 HETERODIMER COMPOSITIONS AND METHODS FOR THE TREATMENT OF OCULAR DISORDERS RIPPLE THERAPEUTICS CORPORATION (CA) 2025-03-06 US disclosed
US-20250057962-A1 PROCESSABLE COMPOSITIONS AND USE FOR THE SAME RIPPLE THERAPEUTICS CORPORATION (CA) 2025-02-20 US disclosed
WO-2023079362-A1 PROCESSABLE COMPOSITIONS AND USE FOR THE SAME RIPPLE THERAPEUTICS CORPORATION (CA) 2023-05-11 WO disclosed
US-11279729-B2 Heterodimer compositions and methods for the treatment of ocular disorders RIPPLE THERAPEUTICS CORPORATION (CA) 2022-03-22 US disclosed
US-20210347809-A1 HETERODIMER COMPOSITIONS AND METHODS FOR THE TREATMENT OF OCULAR DISORDERS RIPPLE THERAPEUTICS CORPORATION (CA) 2021-11-11 US disclosed
US-10822321-B2 Processes and intermediates for the preparations of isomer free prostaglandins CHIROGATE INTERNATIONAL INC. (TW) 2020-11-03 US disclosed
US-10280138-B2 Nitric oxide donating derivatives of fluprostenol NICOX S.A. (FR) 2019-05-07 US disclosed
EP-2349242-B1 AMINO ACID SALTS OF PROSTAGLANDINS NOVAER HOLDINGS INC (US) 2018-12-05 EP disclosed
US-20180251442-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF ISOMER FREE PROSTAGLANDINS CHIROGATE INTERNATIONAL INC. (TW) 2018-09-06 US disclosed
US-20150336921-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF ISOMER FREE PROSTAGLANDINS CHIROGATE INTERNATIONAL INC. (TW) 2015-11-26 US disclosed
US-20150336923-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF ISOMER FREE PROSTAGLANDINS CHIROGATE INTERNATIONAL INC. (TW) 2015-11-26 US disclosed
US-9115109-B2 Processes and intermediates for the preparations of isomer free prostaglandins CHIROGATE INTERNATIONAL INC. (TW) 2015-08-25 US disclosed
US-20150051410-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF ISOMER FREE PROSTAGLANDINS CHIROGATE INTERNATIONAL INC. (TW) 2015-02-19 US disclosed
US-8722739-B2 Amino acid salts of prostaglandins NOVAER HOLDINGS, INC. (US) 2014-05-13 US disclosed
US-8623918-B2 Amino acid salts of prostaglandins NOVAER HOLDINGS, INC. (US) 2014-01-07 US disclosed
US-8470882-B2 2013-06-25 US disclosed
US-20130131106-A1 BIFUNCTIONAL RHO KINASE INHIBITOR COMPOUNDS, COMPOSITION AND USE INSPIRE PHARMACEUTICALS, INC. (US) 2013-05-23 US disclosed
US-20100105771-A1 AMINO ACID SALTS OF PROSTAGLANDINS NOVAER HOLDINGS, INC. 2010-04-29 US disclosed
US-20100105775-A1 AMINO ACID SALTS OF PROSTAGLANDINS NOVAER HOLDINGS, INC. 2010-04-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250074935-A1 HETERODIMER COMPOSITIONS AND METHODS FOR THE TREATMENT OF OCULAR DISORDERS CRYAB, UACA, CRYAA PTGFR 7/4885PTGER3 22/4885ABCC4 4002/4885
US-20250057962-A1 PROCESSABLE COMPOSITIONS AND USE FOR THE SAME CCND2, CCND1, C9 PTGFR 128/4885PTGER3 323/4885ABCC4 2746/4885
US-20180251442-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF ISOMER FREE PROSTAGLANDINS PTGER2, PTGES2, PTGER1 PTGFR 16/4885PTGER3 11/4885ABCC4 2336/4885
US-20100105771-A1 AMINO ACID SALTS OF PROSTAGLANDINS PTGIS, PTGES, PTGIR PTGFR 7/4885PTGER3 16/4885ABCC4 4544/4885
US-20100105775-A1 AMINO ACID SALTS OF PROSTAGLANDINS PTGIS, PTGES, PTGIR PTGFR 7/4885PTGER3 16/4885ABCC4 4544/4885
US-11279729-B2 Heterodimer compositions and methods for the treatment of ocular disorders CRYAB, UACA, CRYAA PTGFR 7/4885PTGER3 22/4885ABCC4 4002/4885
US-20150336923-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF ISOMER FREE PROSTAGLANDINS PTGER2, PTGES2, PTGER1 PTGFR 16/4885PTGER3 11/4885ABCC4 2336/4885
US-10280138-B2 Nitric oxide donating derivatives of fluprostenol PTGIS, NOS2, PTGIR PTGFR 21/4885PTGER3 23/4885ABCC4 2484/4885
US-10822321-B2 Processes and intermediates for the preparations of isomer free prostaglandins PTGER2, PTGES2, PTGER1 PTGFR 16/4885PTGER3 11/4885ABCC4 2336/4885
US-20150336921-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF ISOMER FREE PROSTAGLANDINS PTGER2, PTGES2, PTGER1 PTGFR 16/4885PTGER3 11/4885ABCC4 2336/4885
US-20210347809-A1 HETERODIMER COMPOSITIONS AND METHODS FOR THE TREATMENT OF OCULAR DISORDERS CRYAB, UACA, CRYAA PTGFR 7/4885PTGER3 22/4885ABCC4 4002/4885
US-20150051410-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF ISOMER FREE PROSTAGLANDINS PTGER2, PTGES2, PTGER1 PTGFR 16/4885PTGER3 11/4885ABCC4 2336/4885
US-20130131106-A1 BIFUNCTIONAL RHO KINASE INHIBITOR COMPOUNDS, COMPOSITION AND USE ROCK2, ROCK1, RHOA PTGFR 762/4885PTGER3 1513/4885ABCC4 4340/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.