SCHEMBL3390908

SCHEMBL3390908

COc1cccc(C(=O)N2CCN(c3ccc(NC(=O)N(OS(C)(=O)=O)c4cc(C(C)(C)C)nn4-c4ccc(C)cc4)c(C)n3)CC2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
NAMPT P43490 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
NPY2R P49146 1/20 0.38
CCKAR P32238 3/20 0.37
KMT2A Q03164 1/20 0.37
PTK2B Q14289 1/20 0.37
MAPK14 Q16539 2/20 0.37
PARP14 Q460N5 1/20 0.37
PARP10 Q53GL7 1/20 0.37
BRAF P15056 1/20 0.37
CFTR P13569 1/20 0.36
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3394297 0.93 PTK2B (0.40) ALDH1A1HPGDKMT2APTK2BMAPK14
SCHEMBL3393248 0.93 MAPT (0.43) ALDH1A1CA12CA1CA2CA9
SCHEMBL3392554 0.92 PTK2B (0.37) ALDH1A1CA12CA1CA2CA7
SCHEMBL3393200 0.92 PTK2B (0.37) ALDH1A1NAMPTCA12CA1CA2
SCHEMBL3394251 0.91 PTK2B (0.39) ALDH1A1KMT2APTK2BMAPK14BRAF
SCHEMBL3391076 0.91 PHGDH (0.40) ALDH1A1NPY2RKMT2APTK2BMAPK14
SCHEMBL3392100 0.89 PTK2B (0.39) KMT2APTK2BMAPK14BRAFSRC
SCHEMBL3389398 0.88 PTK2B (0.36) KMT2APTK2BMAPK14BRAFSRC
SCHEMBL3389419 0.88 ALDH1A1 (0.39) ALDH1A1NAMPTNPY2RKMT2APTK2B
SCHEMBL3394286 0.88 LMNA (0.37) ALDH1A1KMT2APTK2BMAPK14BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943243-B1 KINASE INHIBITORS LILLY CO ELI (US) 2010-12-29 EP disclosed