SCHEMBL3394048

SCHEMBL3394048

C=CCOC(=O)CC1(CN)CCCCC1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
TSHR P16473 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
USP2 O75604 1/20 0.51
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
BLM P54132 1/20 0.51
CACNA2D1 P54289 1/20 0.51
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.33
MAPT P10636 1/20 0.33
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33
NPSR1 Q6W5P4 1/20 0.31
CYP3A4 P08684 1/20 0.31
EPHX2 P34913 1/20 0.31
CYP2C19 P33261 1/20 0.31
PKM P14618 1/20 0.31
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL612325 0.98 ALDH1A1 (0.50) ALDH1A1TSHRSMN1; SMN2USP2LMNA
SCHEMBL939773 0.84 ALDH1A1 (0.47) ALDH1A1TSHRSMN1; SMN2USP2LMNA
SCHEMBL7825503 0.80 ALDH1A1 (0.38) ALDH1A1TSHRSMN1; SMN2USP2LMNA
SCHEMBL466295 0.78 ALDH1A1 (0.56) ALDH1A1TSHRSMN1; SMN2USP2LMNA
Hydrochloric Acid SCHEMBL6578159 0.77 ALDH1A1 (0.55) ALDH1A1TSHRSMN1; SMN2USP2LMNA
SCHEMBL14534858 0.75 USP2 (0.62) ALDH1A1TSHRSMN1; SMN2USP2LMNA
SCHEMBL466314 0.75 TSHR (0.62) ALDH1A1TSHRSMN1; SMN2USP2LMNA
SCHEMBL1643330 0.75 TSHR (0.62) ALDH1A1TSHRSMN1; SMN2USP2LMNA
SCHEMBL6545165 0.75 ALDH1A1 (0.38) ALDH1A1TSHRSMN1; SMN2GAATDP1
Hydrochloric Acid SCHEMBL28038690 0.75 ALDH1A1 (0.35) ALDH1A1TSHRSMN1; SMN2USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012164055-A2 NEW COMPOUNDS, SYNTHESIS AND USE THEREOF IN THE TREATMENT OF PAIN LACER, S.A. (ES) 2012-12-06 WO disclosed
EP-2530072-A1 New compounds, synthesis and use thereof in the treatment of pain LACER, S.A. (ES) 2012-12-05 EP disclosed
EP-2172445-A1 Cis (z) 4-t-butylgabapentin and its synthesis Hikal Limited (IN) 2010-04-07 EP disclosed
US-7632864-B2 Gabapentin analogues and process thereof HIKAL LTD. (IN) 2009-12-15 US disclosed
US-20070123591-A1 Gabapentin analogues and process thereof HIKAL LMITED INDIAN INSTITUE OF SCIENCE 2007-05-31 US disclosed
EP-1763503-A1 4-T-BUTYLGABAPENTIN AND ITS SYNTHESIS Hikal Limited (IN) 2007-03-21 EP disclosed
WO-2005087709-A1 4-T-BUTYLGABAPENTIN AND ITS SYNTHESIS HIKAL LIMITED (IN) 2005-09-22 WO disclosed
US-20050209332-A1 Gabapentin analogues and process thereof HIKAL LIMITED 2005-09-22 US disclosed
US-20040063994-A1 Process for the preparation of cyclic amino acids SOLCHEM ITALIANA S.P.A. (IT) 2004-04-01 US disclosed
EP-1373186-A1 A PROCESS FOR THE PREPARATION OF CYCLIC AMINO ACIDS Solchem Italiana S.p.A (IT) 2004-01-02 EP disclosed
WO-2003080588-A1 CYCLIC 1-(ACYLOXY)-ALKYL PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF XENOPORT (US) 2003-10-02 WO disclosed
WO-2002074727-A1 A PROCESS FOR THE PREPARATION OF CYCLIC AMINO ACIDS SOLCHEM ITALIANA S.P.A. (IT) 2002-09-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063994-A1 Process for the preparation of cyclic amino acids SLC7A1, MRPL21, BCAT1 ALDH1A1 2987/4885TSHR 2582/4885SMN1; SMN2 2889/4885
US-20070123591-A1 Gabapentin analogues and process thereof GABRB1, GABRB2, GABRB3 ALDH1A1 1219/4885TSHR 1411/4885SMN1; SMN2 1271/4885
US-20050209332-A1 Gabapentin analogues and process thereof GABRB1, GABRB2, GABRA4 ALDH1A1 1807/4885TSHR 2467/4885SMN1; SMN2 1752/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.