SCHEMBL3405294

SCHEMBL3405294

O=C(Nc1ccccc1)Nc1ccc2c(c1)CCN(C(=O)O)C2

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 11/20 0.63
NPC1 O15118 10/20 0.63
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
SMN1; SMN2 Q16637 3/20 0.58
TP53 P04637 1/20 0.58
TMPRSS2 O15393 4/20 0.58
THRB P10828 1/20 0.52
CASP3 P42574 2/20 0.50
SENP7 Q9BQF6 2/20 0.50
ALDH1A1 P00352 1/20 0.50
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50
TAS1R2 Q8TE23 1/20 0.50
KCNA1 Q09470 1/20 0.50
KCNAB1 Q14722 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
GAA P10253 1/20 0.50
NAMPT P43490 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5459990 0.87 NPC1 (0.67) RAB9ANPC1MEN1KMT2ASMN1; SMN2
SCHEMBL3402909 0.86 NPC1 (0.67) RAB9ANPC1MEN1KMT2ASMN1; SMN2
SCHEMBL5458367 0.84 RAB9A (0.69) RAB9ANPC1MEN1KMT2ASMN1; SMN2
SCHEMBL14862974 0.84 TMPRSS2 (0.61) RAB9ANPC1MEN1KMT2ASMN1; SMN2
SCHEMBL1188540 0.83 ESR2 (0.62) RAB9ANPC1MEN1KMT2ASMN1; SMN2
SCHEMBL5469377 0.83 POLB (0.55) RAB9ANPC1MEN1KMT2ASMN1; SMN2
SCHEMBL5452223 0.83 TMPRSS2 (0.55) RAB9ANPC1MEN1KMT2ATMPRSS2
SCHEMBL3409792 0.81 KCNA1 (0.51) RAB9ANPC1SMN1; SMN2TP53TMPRSS2
SCHEMBL3404203 0.80 THRB (0.49) RAB9ANPC1MEN1KMT2ASMN1; SMN2
SCHEMBL11903038 0.80 TMPRSS2 (0.50) RAB9ANPC1MEN1KMT2ATMPRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2256105-B1 NOVEL TETRAHYDROISOQUINOLINE DERIVATIVE DAIICHI SANKYO CO LTD (JP) 2013-12-04 EP disclosed
EP-2256105-A1 NOVEL TETRAHYDROISOQUINOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2010-12-01 EP disclosed