SCHEMBL3406191

SCHEMBL3406191

COc1cc(Nc2ncc(OC)c(-c3ccccc3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 8/20 0.45
PLK1 P53350 4/20 0.43
KDR P35968 5/20 0.43
CDK1 P06493 4/20 0.43
CSNK1A1 P48729 1/20 0.42
CSNK1D P48730 1/20 0.42
GSK3B P49841 1/20 0.42
CSNK1G2 P78368 1/20 0.42
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3410488 0.82 BRD4 (0.40) IMPDH2PLK1KDRCYP1A2
SCHEMBL3409949 0.82 IMPDH2 (0.51) IMPDH2
SCHEMBL3413376 0.81 GAA (0.43) IMPDH2KDRCDK1MEN1CYP1A2
SCHEMBL3410226 0.81 PLK1 (0.47) PLK1KDRCDK1
SCHEMBL3410455 0.80 MEN1 (0.42) IMPDH2PLK1KDRMEN1CYP1A2
SCHEMBL3412792 0.80 KDR (0.48) PLK1KDRCDK1MAPT
SCHEMBL3410224 0.80 TP53 (0.43) PLK1KDRMEN1MAPTKMT2A
SCHEMBL3413146 0.80 IMPDH2 (0.40) IMPDH2PLK1GSK3B
SCHEMBL3412922 0.80 IMPDH2 (0.39) IMPDH2PLK1
SCHEMBL3408743 0.80 PRKCA (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed