SCHEMBL3431063

SCHEMBL3431063

CC(C)(C)c1nc2c(CCC(=O)O)cc(-c3ccc(Cl)c(C(F)(F)F)c3)cc2[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
GALK1 P51570 1/20 0.39
CDK8 P49336 1/20 0.37
PTGES O14684 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
COMT P21964 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
SLC22A12 Q96S37 1/20 0.35
GCGR P47871 3/20 0.34
NOTUM Q6P988 4/20 0.34
CYP1A2 P05177 1/20 0.34
GPR17 Q13304 1/20 0.34
PRKCZ Q05513 1/20 0.34
ABL1 P00519 1/20 0.34
BCR P11274 1/20 0.34
SRC P12931 1/20 0.34
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346903 0.90 GRIN2B (0.36) PDE3BPDE3AGCGRFFAR4
SCHEMBL3346289 0.85 PDE5A (0.40) PTGESGCGRFFAR4
SCHEMBL3346056 0.84 S1PR1 (0.41) GPR17
SCHEMBL3346086 0.82 PTGER4 (0.44) CYP2C9GPR17
SCHEMBL3347691 0.78 FFAR4 (0.40) FFAR4
SCHEMBL3430892 0.76 FFAR4 (0.44) CYP2C9FFAR4
SCHEMBL3431483 0.74 FFAR1 (0.43) GCGRFFAR4
SCHEMBL3350657 0.69 DHODH (0.41) CYP3A4CYP2C9CYP1A2CHEK2
SCHEMBL3430044 0.68 FFAR1 (0.48) GCGRFFAR4
SCHEMBL3352922 0.68 GSK3B (0.38) PTGESCYP2C9GCGRFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010053757-A1 2 -OXOQUINOXALIN BLOCKERS OF THE LATE SODIUM CHANNEL GILEAD PALO ALTO, INC. (US) 2010-05-14 WO disclosed