SCHEMBL3432976

SCHEMBL3432976

CC(=O)OCC(=O)NCCc1cc(-c2ccc(OC(F)(F)F)cc2)cc2[nH]c(=O)c(C(F)(F)F)nc12

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.39
KDM4E B2RXH2 4/20 0.37
HSD17B10 Q99714 4/20 0.37
TRPV1 Q8NER1 10/20 0.36
TSHR P16473 2/20 0.36
HPGD P15428 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
P2RY12 Q9H244 1/20 0.34
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
PABPC1 P11940 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3430772 0.78 KDM4E (0.38) GSK3BKDM4EHSD17B10TRPV1TSHR
SCHEMBL3346362 0.75 DHODH (0.39) KDM4EHSD17B10TRPV1TSHRALDH1A1
SCHEMBL3344258 0.71 KDM4E (0.43) GSK3BKDM4EHSD17B10TRPV1TSHR
SCHEMBL3475197 0.70 SCD (0.47)
SCHEMBL3430136 0.70 DHODH (0.39) KDM4EHSD17B10TRPV1HPGDMAPT
SCHEMBL3352922 0.70 GSK3B (0.38) GSK3B
SCHEMBL3352967 0.69 NR1D1 (0.40) GSK3BKDM4EHSD17B10TRPV1TSHR
SCHEMBL3428421 0.69 PPARD (0.39) GSK3B
SCHEMBL3430623 0.67 FFAR1 (0.43) KDM4EHSD17B10HPGDALDH1A1
SCHEMBL4493825 0.66 GSK3B (0.78) GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010053757-A1 2 -OXOQUINOXALIN BLOCKERS OF THE LATE SODIUM CHANNEL GILEAD PALO ALTO, INC. (US) 2010-05-14 WO claimed