SCHEMBL3468280

SCHEMBL3468280

COC(=O)C(CCc1ccc(-c2cccc(C#N)c2)cc1)Cc1ccc(Br)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 2/20 0.53
MMP13 P45452 2/20 0.53
MME P08473 2/20 0.46
CTSC P53634 2/20 0.44
HDAC1 Q13547 6/20 0.40
HDAC6 Q9UBN7 6/20 0.40
ADAMTS4 O75173 1/20 0.39
MCHR1 Q99705 1/20 0.39
NLRP3 Q96P20 1/20 0.38
FFAR1 O14842 2/20 0.38
FFAR4 Q5NUL3 1/20 0.38
FOLH1 Q04609 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3467200 0.87 MMP12 (0.60) MMP12MMP13MMECTSCADAMTS4
SCHEMBL3466565 0.85 GPR34 (0.54) MMP12MMP13ADAMTS4FFAR1FFAR4
SCHEMBL3467017 0.82 MMP12 (0.57) MMP12MMP13MMEADAMTS4MCHR1
SCHEMBL7924636 0.80 MMP12 (0.65) MMP12MMP13MMECTSCADAMTS4
SCHEMBL3467000 0.77 MMP12 (0.51) MMP12MMP13ADAMTS4FFAR1FFAR4
SCHEMBL3467425 0.76 MMP12 (0.54) MMP12MMP13MMECTSCADAMTS4
SCHEMBL3466777 0.76 MMP12 (0.54) MMP12MMP13MMECTSCADAMTS4
SCHEMBL3466325 0.75 FFAR1 (0.57) MMP12MMP13ADAMTS4FFAR1FFAR4
SCHEMBL12646553 0.74 MMP12 (0.56) MMP12MMP13MMEHDAC1ADAMTS4
SCHEMBL7928277 0.73 MMP12 (0.64) MMP12MMP13MMEADAMTS4FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010070076-A1 ALKANOIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE AS HDAC INHIBITORS CRYSTAX PHARMACEUTICALS, S.L. (ES) 2010-06-24 WO claimed
WO-2010070076-A1 ALKANOIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE AS HDAC INHIBITORS CRYSTAX PHARMACEUTICALS, S.L. (ES) 2010-06-24 WO disclosed