Water

Water

SCHEMBL3478298

C=CCNCc1ccccc1.O

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 1/20 0.54
CHRM2 known ✓ P08172 1/20 0.47
SIGMAR1 known ✓ Q99720 1/20 0.44
THRB known ✓ P10828 1/20 0.43
KMT2A Q03164 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
DPP7 Q9UHL4 1/20 0.52
ADH1B P00325 1/20 0.48
ADH1C P00326 1/20 0.48
ADH1A P07327 1/20 0.48
ADH7 P40394 1/20 0.48
MAOA P21397 1/20 0.48
MAPT P10636 2/20 0.47
GAA P10253 2/20 0.47
KDM4E B2RXH2 2/20 0.46
CYP3A4 P08684 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 1/20 0.44
IDO1 P14902 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681149 0.98 MEN1 (0.56) MEN1KMT2ATDP1DPP7ADH1B
Ammonia Solution, Strong SCHEMBL27753398 0.96 MEN1 (0.54) MEN1KMT2ATDP1DPP7ADH1B
Hydrochloric Acid SCHEMBL250190 0.96 MEN1 (0.54) MEN1KMT2ATDP1DPP7ADH1B
Bromide SCHEMBL9394202 0.96 MEN1 (0.54) MEN1KMT2ATDP1DPP7ADH1B
Hypochlorous Acid SCHEMBL28117107 0.90 MEN1 (0.48) MEN1KMT2ATDP1DPP7ADH1B
Oxalic Acid SCHEMBL29028526 0.88 KDM4E (0.57) MEN1KMT2ATDP1DPP7ADH1B
Phenol SCHEMBL28870632 0.88 MEN1 (0.47) MEN1KMT2ATDP1DPP7ADH1B
SCHEMBL17291833 0.86 DPP7 (0.44) MEN1KMT2ATDP1DPP7ADH1B
Phenethylamine SCHEMBL8068653 0.85 HTR2A (0.55) MEN1KMT2ATDP1DPP7ADH1B
SCHEMBL366586 0.83 CHRM2 (0.40) MEN1KMT2ATDP1DPP7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119430216-A Titanium-silicon molecular sieve and preparation method and application thereof 中国石油化工股份有限公司 2025-02-14 CN claimed
CN-119430216-A Titanium-silicon molecular sieve and preparation method and application thereof 中国石油化工股份有限公司 2025-02-14 CN disclosed
CN-106164035-B Biomass treatment process 英国萨培生物科技有限公司 2020-01-07 CN disclosed
US-10174131-B2 Biomass processing method SAPPI BIOTECH UK LTD (GB) 2019-01-08 US disclosed
WO-2018154314-A1 HEMICELLULOSE PROCESSING METHOD SAPPI BIOTECH UK LIMITED (GB) 2018-08-30 WO disclosed
EP-3129346-A1 BIOMASS PROCESSING METHOD Plaxica Limited (GB) 2017-02-15 EP disclosed
US-20170029532-A1 BIOMASS PROCESSING METHOD PLAXICA LIMITED (GB) 2017-02-02 US disclosed
WO-2015155534-A1 BIOMASS PROCESSING METHOD PLAXICA LIMITED (GB) 2015-10-15 WO disclosed
EP-1907445-B1 AMINE AQUEOUS SOLUTION FOR FORMING AN ACTIVE LAYER OF POLYAMIDE REVERSE OSMOSIS COMPOSITE MEMBRANE AND PREPARATION METHOD OF POLYAMIDE REVERSE OSMOSIS COMPOSITE MEMBRANE USING THE SAME WOONGJINCOWAY CO LTD (KR) 2013-03-13 EP disclosed
WO-2012131299-A1 PROCESS FOR PRODUCING LACTATE PLAXICA LIMITED (GB) 2012-10-04 WO disclosed
US-7766173-B2 Polyamide reverse osmosis composite membrane and preparation method thereof WOONGJINCOWAY CO., LTD. (KR) 2010-08-03 US disclosed
US-20080237118-A1 Polyamide Reverse Osmosis Composite Membrane and Preparation Method Thereof WOONGJINCOWAY CO. LTD. (KR) 2008-10-02 US disclosed
EP-1907445-A1 POLYAMIDE REVERSE OSMOSIS COMPOSITE MEMBRANE AND PREPARATION METHOD THEREOF Woongjincoway Co, Ltd. (KR) 2008-04-09 EP disclosed
WO-2007013710-A1 POLYAMIDE REVERSE OSMOSIS COMPOSITE MEMBRANE AND PREPARATION METHOD THEREOF WOONGJINCOWAY CO, LTD,. (KR) 2007-02-01 WO disclosed
US-5502195-A Sulfoxide-carboxylate intermediates of omeprazole and lansoprazole TORCAN CHEMICAL LTD. (CA) 1996-03-26 US disclosed