SCHEMBL3572023

SCHEMBL3572023

CC1OC(=O)N(c2ccccc2)C1(O)N1CCC(F)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.35
ALDH1A1 P00352 4/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD11B1 P28845 5/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPC1 O15118 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ATM Q13315 1/20 0.32
IDH1 O75874 2/20 0.31
FADS1 O60427 1/20 0.31
POLB P06746 1/20 0.31
DRD2 P14416 1/20 0.30
DRD4 P21917 1/20 0.30
DRD3 P35462 1/20 0.30
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3570224 0.68 ALDH1A1 (0.33) ALDH1A1CYP2C19KDM4EHPGDL3MBTL1
SCHEMBL7668531 0.67 HTT (0.38) MAOAALDH1A1KDM4EL3MBTL1IDH1
SCHEMBL3578041 0.65 OPRM1 (0.32) MAOADRD2DRD3
SCHEMBL3576644 0.65 HSD11B1 (0.37) ALDH1A1CYP1A2CYP2C9CYP2C19HSD11B1
Methane SCHEMBL3572022 0.62 ALDH1A1 (0.38) ALDH1A1CYP1A2CYP2C9CYP2C19HSD11B1
SCHEMBL3618028 0.61 ALDH1A1 (0.37) ALDH1A1CYP1A2CYP2C9CYP2C19HSD11B1
SCHEMBL3575081 0.59 ALDH1A1 (0.40) MAOAALDH1A1KDM4EHPGDL3MBTL1
SCHEMBL4477880 0.59 MBTD1 (0.59) ALDH1A1CYP2C9CYP2C19SMN1; SMN2L3MBTL1
SCHEMBL9731036 0.59 MAOA (0.43) MAOAALDH1A1KDM4EHPGDRAB9A
SCHEMBL7812799 0.58 ALDH1A1 (0.35) ALDH1A1CYP1A2CYP2C9CYP2C19HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8729269-B2 Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy WOCKHARDT LIMITED (IN) 2014-05-20 US disclosed
US-20100144735-A1 SUBSTITUTED PIPERIDINO PHENYLOXAZOLIDINONES HAVING ANTIMICROBIAL ACTIVITY WITH IMPROVED IN VIVO EFFICACY WOCKHARDT LIMITED 2010-06-10 US disclosed
US-7687627-B2 Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy WOCKHARDT LIMITED (IN) 2010-03-30 US disclosed
EP-1664038-A2 SUBSTITUTED PIPERIDINO PHENYLOXAZOLIDINONES HAVING ANTIMICRIOBIAL ACTIVITY WITH IMPROVED I IN VIVO /I EFFICACY Wockhardt Limited (IN) 2006-06-07 EP disclosed
US-20050143421-A1 Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy WOCKHARDT LIMITED 2005-06-30 US disclosed
WO-2005054234-A2 SUBSTITUTED PIPERIDINO PHENYLOXAZOLIDINONES HAVING ANTIMICRIOBIAL ACTIVITY WITH IMPROVED IN VIVO EFFICACY WOCKHARDT LIMITED (IN) 2005-06-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100144735-A1 SUBSTITUTED PIPERIDINO PHENYLOXAZOLIDINONES HAVING ANTIMICROBIAL ACTIVITY WITH IMPROVED IN VIVO EFFICACY GMPS, MPO, ARG1 MAOA 2638/4885ALDH1A1 1960/4885CYP1A2 2277/4885
US-20050143421-A1 Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy GMPS, MPO, ARG1 MAOA 2638/4885ALDH1A1 1960/4885CYP1A2 2277/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.