SCHEMBL3574044

SCHEMBL3574044

CNc1cnc(Cl)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(C)(C)C)cc1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.37
CCR9 P51686 2/20 0.37
ESRRG P62508 2/20 0.36
ESRRB O95718 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
HSP90AA1 P07900 2/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
NR1I3 Q14994 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.33
VNN1 O95497 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580029 0.90 MLYCD (0.34) SIGMAR1HSP90AA1OPRM1OPRD1
SCHEMBL1397709 0.89 OPRM1 (0.35) CCR9SIGMAR1OPRM1OPRD1
SCHEMBL3574429 0.88 KDM4C (0.39) NR1H4ESRRGESRRBSIGMAR1HSP90AA1
SCHEMBL3579370 0.87 SLC2A1 (0.39) TRPM8
SCHEMBL3571051 0.86 NR1H4 (0.37) NR1H4ESRRGESRRBSIGMAR1HSP90AA1
SCHEMBL3579634 0.86 SERPINE1 (0.40) NR1H4CCR9ESRRGESRRBSIGMAR1
SCHEMBL12520875 0.85 TRPM8 (0.40) NR1H4CCR9ESRRGESRRBOPRM1
SCHEMBL3575452 0.85 KMT2A (0.42) NR1H4ESRRGESRRBSIGMAR1HSP90AA1
SCHEMBL3584245 0.84 SIGMAR1 (0.34) SIGMAR1OPRM1OPRD1
SCHEMBL3576692 0.83 ESRRG (0.37) NR1H4CCR9ESRRGESRRBSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed