SCHEMBL3583661

SCHEMBL3583661

CC(C)(C)c1ccc(CN(CCc2ccc(Cl)c(Cl)c2)C(=O)c2cccnc2NC2CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 3/20 0.41
CRHR1 P34998 3/20 0.37
RAF1 P04049 1/20 0.36
MAP2K1 Q02750 1/20 0.36
P2RX7 Q99572 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TRPV1 Q8NER1 2/20 0.35
NR1H4 Q96RI1 1/20 0.34
ESRRB O95718 1/20 0.34
ESRRG P62508 1/20 0.34
TRPA1 O75762 1/20 0.33
KCNH2 Q12809 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580658 0.89 RAF1 (0.39) RAF1MAP2K1OPRM1OPRD1MEN1
SCHEMBL3580209 0.88 MCHR1 (0.40) BTKCRHR1HDAC3HDAC8HDAC6
SCHEMBL3576972 0.87 BTK (0.36) BTKCRHR1HDAC3HDAC8HDAC6
SCHEMBL3581747 0.85 CCR9 (0.39) RAF1MAP2K1OPRM1OPRD1MEN1
SCHEMBL3573203 0.84 RAF1 (0.40) RAF1MAP2K1OPRM1OPRD1MEN1
SCHEMBL3582883 0.83 RAF1 (0.40) RAF1MAP2K1OPRM1OPRD1MEN1
SCHEMBL3572867 0.82 MEN1 (0.38) HDAC3HDAC8HDAC6OPRM1OPRD1
SCHEMBL3575452 0.81 KMT2A (0.42) RAF1MAP2K1OPRM1OPRD1MEN1
SCHEMBL3581464 0.80 TRPV1 (0.41) RAF1MAP2K1OPRM1OPRD1MEN1
SCHEMBL3580336 0.80 MAPT (0.42) RAF1MAP2K1OPRM1OPRD1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed