SCHEMBL3586516

SCHEMBL3586516

Nc1ccc(C(=O)NN[C@@H](CCC(=O)O)C(=O)O)c([N+](=O)[O-])c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
CYP3A4 P08684 4/20 0.40
ALOX15 P16050 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
TYMS P04818 2/20 0.40
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CA2 P00918 2/20 0.38
CA1 P00915 1/20 0.38
HPGD P15428 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CTSD P07339 1/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 2/20 0.36
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3572326 0.94 TYMS (0.39) ALDH1A1CYP3A4ALOX15TDP1TYMS
SCHEMBL3572332 0.84 CYP3A4 (0.33) ALDH1A1CYP3A4ALOX15TDP1TYMS
SCHEMBL3634693 0.81 MAPT (0.40) ALDH1A1CYP3A4ALOX15TDP1MAPK1
SCHEMBL3574966 0.77 ITGA4 (0.35) ALDH1A1CYP3A4ALOX15TDP1MAPK1
Trifluoroacetic Acid SCHEMBL3585015 0.77 MAPT (0.36) ALDH1A1CYP3A4ALOX15TDP1TYMS
SCHEMBL21422767 0.73 MAPT (0.37) ALDH1A1CYP3A4ALOX15TDP1TYMS
SCHEMBL5925568 0.72 CA2 (0.52) ALDH1A1CYP3A4TDP1CA2CA1
SCHEMBL9828354 0.71 CTSD (0.55) ALDH1A1CYP3A4TYMSCA2CA1
SCHEMBL27456509 0.71 CTSD (0.55) ALDH1A1CYP3A4TYMSCA2CA1
SCHEMBL28907592 0.70 DHFR (0.53) ALDH1A1TYMSCA2CA1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150514-B1 18F-LABELLED FOLATES Merck & Cie (CH) 2018-10-24 EP disclosed
US-9771368-B2 18F-labelled folates Merck & Cie (CH) 2017-09-26 US disclosed
US-20160159802-A1 18F-LABELLED FOLATES Merck & Cie (CH) 2016-06-09 US disclosed
US-9315506-B2 18F-labelled folates Merck & Cie (CH) 2016-04-19 US disclosed
US-20100056533-A1 18F-LABELLED FOLATES MERCK EPROVA AG (CH) 2010-03-04 US disclosed
EP-2150514-A2 18F-LABELLED FOLATES Merck Eprova AG (CH) 2010-02-10 EP disclosed
CN-101646670-A 18F-labelled folates MERCK EPROVA AG CH 2010-02-10 CN disclosed
WO-2008125617-A2 18F-LABELLED FOLATES MERCK EPROVA AG (CH) 2008-10-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056533-A1 18F-LABELLED FOLATES FOLR1, FOLR2, SLC19A1 ALDH1A1 1012/4885CYP3A4 1686/4885ALOX15 996/4885
US-20160159802-A1 18F-LABELLED FOLATES FOLR1, FOLR2, SLC19A1 ALDH1A1 942/4885CYP3A4 2092/4885ALOX15 835/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.