SCHEMBL3609202

SCHEMBL3609202

CCCCCN1CCc2ccccc2C1C(=O)Nc1cc(C)c(OC(C)=O)c(C)c1C

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 3/20 0.42
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
OPRM1 P35372 2/20 0.41
OPRK1 P41145 2/20 0.41
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
HDAC1 Q13547 3/20 0.36
HDAC2 Q92769 3/20 0.36
HDAC8 Q9BY41 3/20 0.36
HDAC3 O15379 2/20 0.36
NCOR2 Q9Y618 2/20 0.36
DRD2 P14416 3/20 0.36
DRD1 P21728 3/20 0.36
HTR2A P28223 2/20 0.35
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3608890 0.87 OPRM1 (0.44) PPARDPPARGPPARAOPRM1OPRK1
SCHEMBL3609022 0.86 PPARD (0.43) PPARDPPARGPPARAOPRM1OPRK1
Hydrochloric Acid SCHEMBL3606029 0.86 OPRM1 (0.44) PPARDPPARGPPARAOPRM1OPRK1
SCHEMBL3604131 0.81 DRD2 (0.37) PPARDPPARGPPARADRD2DRD1
SCHEMBL3606227 0.79 PPARD (0.46) PPARDPPARGPPARA
Hydrochloric Acid SCHEMBL3602849 0.76 RORC (0.36)
SCHEMBL3605281 0.75 GHSR (0.47)
SCHEMBL3614097 0.74 RORC (0.37)
SCHEMBL3612271 0.74 KMT2A (0.36)
SCHEMBL3607481 0.73 TMEM97 (0.37) DRD1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100022582-A1 Tetrahydroisoquinoline Compound and Medicinal Use Thereof KYOTO PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2010-01-28 US disclosed
EP-1857444-A1 TETRAHYDROISOQUINOLINE COMPOUND AND MEDICINAL USE THEREOF Kyoto Pharmaceutical Industries, Ltd. (JP) 2007-11-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100022582-A1 Tetrahydroisoquinoline Compound and Medicinal Use Thereof ACAT1, ACAT2, LCAT PPARD 805/4885PPARG 443/4885PPARA 542/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.